Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50043009
TargetOrexin receptor type 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50434481(CHEMBL2385133 | CHEMBL2385134 | CHEMBL2385132)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at OX2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50434481(CHEMBL2385133 | CHEMBL2385134 | CHEMBL2385132)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at OX1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin receptor type 2(Human)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50434481(CHEMBL2385133 | CHEMBL2385134 | CHEMBL2385132)
Affinity DataKi:  1.10nMAssay Description:Antagonist activity at OX2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)