Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50042924
TargetSphingosine kinase 1(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50433311(CHEMBL2376444)
Affinity DataEC50:  8.30E+3nMAssay Description:Activation of recombinant GFP-tagged SK1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins by Cerenkov counting...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine kinase 1(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50433312(CHEMBL2376443)
Affinity DataEC50:  5.70E+3nMAssay Description:Activation of recombinant GFP-tagged SK1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins by Cerenkov counting...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSphingosine kinase 1(Human)
The City University of New York

Curated by ChEMBL
LigandPNGBDBM50004888(CHEMBL1773676 | (S)-Fingolimod Vinylphosphonate)
Affinity DataKi:  1.00E+4nMAssay Description:Competitive inhibition of SK1 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed