Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50042781
TargetAndrogen receptor(Mouse)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Mouse)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430945(CHEMBL2336987)
Affinity DataIC50: 460nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430946(CHEMBL2336980)
Affinity DataIC50: 990nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430944(CHEMBL2336966)
Affinity DataIC50: 1.46E+3nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430944(CHEMBL2336966)
Affinity DataIC50: 4.45E+3nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430946(CHEMBL2336980)
Affinity DataIC50: 2.56E+4nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Mouse)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430945(CHEMBL2336987)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed