Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50042937
TargetSerine/threonine-protein kinase PLK1(Human)
Korea Basic Science Institute

Curated by ChEMBL
LigandPNGBDBM50433414(CHEMBL2380650)
Affinity DataIC50: 120nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Korea Basic Science Institute

Curated by ChEMBL
LigandPNGBDBM50433415(CHEMBL2380764)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Korea Basic Science Institute

Curated by ChEMBL
LigandPNGBDBM50433416(CHEMBL2380660)
Affinity DataIC50: 2.56E+3nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Korea Basic Science Institute

Curated by ChEMBL
LigandPNGBDBM50433413(CHEMBL2380651)
Affinity DataIC50: 4.75E+3nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Korea Basic Science Institute

Curated by ChEMBL
LigandPNGBDBM50433417(CHEMBL2380653)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Korea Basic Science Institute

Curated by ChEMBL
LigandPNGBDBM50433418(CHEMBL2380765)
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Korea Basic Science Institute

Curated by ChEMBL
LigandPNGBDBM50426931(CHEMBL2323729 | US20230365568, Compound 6a)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of HA-EGFP tagged Plk1 polo-box domain (unknown origin) expressed in 293A cells assessed as inhibition of biotin-p-T78 binding after 1 hr ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed