Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50042517
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 1.40nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 4.90nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 6.70nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Human)
College of Pharmacy of Kangwon National University
Curated by ChEMBL
College of Pharmacy of Kangwon National University
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at human GPR119 transfected in HEK293 cells assessed as concentration for 50 % cAMP stimulation of oleylethanolamineMore data for this Ligand-Target Pair
