Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50042669
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429094(CHEMBL2335783)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli using 2- thio-PAF as substrate incubated for 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429098(CHEMBL2335784)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli using 2- thio-PAF as substrate incubated for 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429070(CHEMBL2335742)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli using 2- thio-PAF as substrate incubated for 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429101(CHEMBL2335780)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli using 2- thio-PAF as substrate incubated for 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429098(CHEMBL2335784)
Affinity DataIC50: 9nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429070(CHEMBL2335742)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hr in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429101(CHEMBL2335780)
Affinity DataIC50: 10nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429094(CHEMBL2335783)
Affinity DataIC50: 10nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429114(CHEMBL2335769)
Affinity DataIC50: 13nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429113(CHEMBL2335770)
Affinity DataIC50: 14nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429112(CHEMBL2335760)
Affinity DataIC50: 16nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429070(CHEMBL2335742)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli using 2- thio-PAF as substrate incubated for 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429111(CHEMBL2335786)
Affinity DataIC50: 22nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429110(CHEMBL2335749)
Affinity DataIC50: 23nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429108(CHEMBL2335779)
Affinity DataIC50: 26nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429109(CHEMBL2335768)
Affinity DataIC50: 26nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429070(CHEMBL2335742)
Affinity DataIC50: 27nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429107(CHEMBL2335782)
Affinity DataIC50: 28nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429106(CHEMBL2335767)
Affinity DataIC50: 31nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429105(CHEMBL2335748)
Affinity DataIC50: 32nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429078(CHEMBL2335755)
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli using 2- thio-PAF as substrate incubated for 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429104(CHEMBL2335747)
Affinity DataIC50: 38nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429102(CHEMBL2335778)
Affinity DataIC50: 39nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429103(CHEMBL2335771)
Affinity DataIC50: 39nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429101(CHEMBL2335780)
Affinity DataIC50: 41nMAssay Description:Inhibition of TAMRA-tagged AX4870 labeling of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli incubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429070(CHEMBL2335742)
Affinity DataIC50: 42nMAssay Description:Inhibition of TAMRA-tagged AX4870 labeling of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli incubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429100(CHEMBL2335763)
Affinity DataIC50: 44nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429070(CHEMBL2335742)
Affinity DataIC50: 46nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hr in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429099(CHEMBL2335772)
Affinity DataIC50: 49nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429098(CHEMBL2335784)
Affinity DataIC50: 49nMAssay Description:Inhibition of TAMRA-tagged AX4870 labeling of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli incubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429097(CHEMBL2335773)
Affinity DataIC50: 52nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429096(CHEMBL2335746)
Affinity DataIC50: 55nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429095(CHEMBL2335781)
Affinity DataIC50: 55nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429094(CHEMBL2335783)
Affinity DataIC50: 59nMAssay Description:Inhibition of TAMRA-tagged AX4870 labeling of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli incubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429093(CHEMBL2335761)
Affinity DataIC50: 70nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429092(CHEMBL2335785)
Affinity DataIC50: 80nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429091(CHEMBL2335762)
Affinity DataIC50: 87nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429089(CHEMBL2335757)
Affinity DataIC50: 100nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429088(CHEMBL2335777)
Affinity DataIC50: 100nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429087(CHEMBL2335774)
Affinity DataIC50: 120nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429086(CHEMBL2335758)
Affinity DataIC50: 150nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429085(CHEMBL2335759)
Affinity DataIC50: 150nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429078(CHEMBL2335755)
Affinity DataIC50: 170nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429084(CHEMBL2335745)
Affinity DataIC50: 230nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429083(CHEMBL2335764)
Affinity DataIC50: 240nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429082(CHEMBL2335775)
Affinity DataIC50: 250nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429081(CHEMBL2335751)
Affinity DataIC50: 370nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429080(CHEMBL2335776)
Affinity DataIC50: 450nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429079(CHEMBL2335753)
Affinity DataIC50: 820nMAssay Description:Inhibition of human plasma Lp-PLA2 using 2- thio-PAF as substrate incubated for 20 mins prior to substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50429078(CHEMBL2335755)
Affinity DataIC50: 830nMAssay Description:Inhibition of TAMRA-tagged AX4870 labeling of human recombinant N-terminal hexahistidine-tagged Lp-PLA2 expressed in Escherichia coli incubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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