Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50040821
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400690(CHEMBL2203524)
Affinity DataIC50: 7nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400689(CHEMBL2203525)
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400664(CHEMBL2204239)
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400684(CHEMBL2203528)
Affinity DataIC50: 76nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400662(CHEMBL2204241)
Affinity DataIC50: 78nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400665(CHEMBL2204238)
Affinity DataIC50: 110nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400682(CHEMBL2203530)
Affinity DataIC50: 150nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400668(CHEMBL2204235)
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400687(CHEMBL1992679)
Affinity DataIC50: 170nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400666(CHEMBL2204237)
Affinity DataIC50: 250nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400663(CHEMBL2204240)
Affinity DataIC50: 270nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM67675(N-[2-(3-oxo-4H-quinoxalin-2-yl)phenyl]-2-thiophene...)
Affinity DataIC50: 280nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400681(CHEMBL2203531)
Affinity DataIC50: 300nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400686(CHEMBL2203526)
Affinity DataIC50: 380nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400667(CHEMBL2204236)
Affinity DataIC50: 410nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400685(CHEMBL2203527)
Affinity DataIC50: 530nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400683(CHEMBL2203529)
Affinity DataIC50: 580nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400680(CHEMBL2203532)
Affinity DataIC50: 980nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400669(CHEMBL2204234)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400676(CHEMBL2203536)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400670(CHEMBL2204233)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400671(CHEMBL2204232)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400672(CHEMBL2204231)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400673(CHEMBL2204230)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400679(CHEMBL2203533)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400678(CHEMBL2203534)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400677(CHEMBL2203535)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400675(CHEMBL2204228)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 33(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400674(CHEMBL2204229)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal 6His-tagged full length human recombinant STK33 using myelin basic protein as substrate incubated for 15 mins before initiat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed