Compile Data Set for Download or QSAR
Report error Found 132 Enz. Inhib. hit(s) with all data for entry = 50040733
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399112(CHEMBL2179776)
Affinity DataEC50:  159nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399121(CHEMBL2179751)
Affinity DataEC50:  28.3nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399119(CHEMBL2179754)
Affinity DataEC50:  17.1nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataEC50:  13.7nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399122(CHEMBL2179734)
Affinity DataEC50:  13.4nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399120(CHEMBL2179771)
Affinity DataEC50:  5.73nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399118(CHEMBL2179763)
Affinity DataEC50:  4.11nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399157(CHEMBL2179724)
Affinity DataEC50:  83.8nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as reduction in forskolin-induced cAMP accumulation incubated for 45 mins by T...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  10.6nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399121(CHEMBL2179751)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399121(CHEMBL2179751)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399122(CHEMBL2179734)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399122(CHEMBL2179734)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399120(CHEMBL2179771)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399120(CHEMBL2179771)
Affinity DataKi:  64nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399119(CHEMBL2179754)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399119(CHEMBL2179754)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399118(CHEMBL2179763)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399118(CHEMBL2179763)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399117(CHEMBL2179740)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399117(CHEMBL2179740)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399116(CHEMBL2179762)
Affinity DataKi:  109nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399115(CHEMBL2179735)
Affinity DataKi:  146nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399115(CHEMBL2179735)
Affinity DataKi:  146nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399114(CHEMBL2179759)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399114(CHEMBL2179759)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399113(CHEMBL2179739)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399113(CHEMBL2179739)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399111(CHEMBL2179736)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399111(CHEMBL2179736)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399110(CHEMBL2179728)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399110(CHEMBL2179728)
Affinity DataKi:  167nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399109(CHEMBL2179733)
Affinity DataKi:  182nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399109(CHEMBL2179733)
Affinity DataKi:  182nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399108(CHEMBL2179753)
Affinity DataKi:  203nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399108(CHEMBL2179753)
Affinity DataKi:  203nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399107(CHEMBL2179727)
Affinity DataKi:  213nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399107(CHEMBL2179727)
Affinity DataKi:  213nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399106(CHEMBL2179752)
Affinity DataKi:  221nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399106(CHEMBL2179752)
Affinity DataKi:  221nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399105(CHEMBL2179738)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399105(CHEMBL2179738)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399123(CHEMBL2179766)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399123(CHEMBL2179766)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399124(CHEMBL2179737)
Affinity DataKi:  462nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399124(CHEMBL2179737)
Affinity DataKi:  462nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399116(CHEMBL2179762)
Affinity DataKi:  494nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399116(CHEMBL2179762)
Affinity DataKi:  494nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399125(CHEMBL2179755)
Affinity DataKi:  595nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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