Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50040578
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50396334(CHEMBL2170034)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]chloroquine uptake...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50396333(CHEMBL2170036)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]chloroquine uptake...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM519(SQV | Invirase | CHEMBL114 | Ro 31-8959 | Fortovas...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]chloroquine uptake...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetChloroquine resistance transporter(malaria parasite P. falciparum)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50338982((R)-5-((3,4-dimethoxyphenethyl)(methyl)amino)-2-(3...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocyte assessed as inhibition of [3H]chloroquine uptake...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed