Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50040019
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50: 300nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of MEK2 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387975(CHEMBL2057831)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387975(CHEMBL2057831)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM14800(2-(5,6-Diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-et...)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387976(CHEMBL2057832)
Affinity DataIC50: 2.31E+4nMAssay Description:Inhibition of MEK1 using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM14800(2-(5,6-Diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-et...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50387976(CHEMBL2057832)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of PI3Kalpha using [gamma32P]ATP by radiometric kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed