Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50039986
Affinity DataIC50: 5nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 165nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 229nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of FYNMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ITKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of LYNMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ZAP70More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ERK1More data for this Ligand-Target Pair
TargetRAF proto-oncogene serine/threonine-protein kinase(Human)
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of c-RafMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of PKCtheta-mediated IL-2 production by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of PKCepsilonMore data for this Ligand-Target Pair
