Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50040491
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50: 11nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50: 14nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50: 23nMAssay Description:Inhibition of UT-B-mediated urea transport in wild type CD1 mouse erythrocytes incubated for 10 mins prior to urea addition by Stopped-flow light sca...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50: 25.1nMAssay Description:Reversible inhibition of mouse UT-B-mediated urea transportMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394964(CHEMBL1590659)
Affinity DataIC50: 32nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394967(CHEMBL2165784)
Affinity DataIC50: 104nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394972(CHEMBL1372659)
Affinity DataIC50: 153nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394966(CHEMBL2165785)
Affinity DataIC50: 196nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50322183(CHEMBL1173569 | UT-A1 inhibitor D4 | 3-(4-ethylphe...)
Affinity DataIC50: 212nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394965(CHEMBL2165786)
Affinity DataIC50: 468nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394970(CHEMBL2165781)
Affinity DataIC50: 537nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394969(CHEMBL2165782)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394963(CHEMBL2165787)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394968(CHEMBL2165783)
Affinity DataIC50: 5.29E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394974(CHEMBL1725922)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394971(CHEMBL2165780)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394973(CHEMBL2165789)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed