Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 5615
TargetSerine/threonine-protein kinase PLK1(Human)
Frederick National Laboratory For Cancer Research

LigandPNGBDBM91675(Peptide-peptoid hybrid, 6q)
Affinity DataIC50: 15nMAssay Description:Pkk1 PDB fluorescence polarization competition binding assay using Plk. More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Frederick National Laboratory For Cancer Research

LigandPNGBDBM91676(Peptide-peptoid hybrid, 7)
Affinity DataIC50: 19nMAssay Description:Pkk1 PDB fluorescence polarization competition binding assay using Plk. More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Frederick National Laboratory For Cancer Research

LigandPNGBDBM91677(Peptide-peptoid hybrid, 13)
Affinity DataIC50: 71nMAssay Description:Pkk1 PDB fluorescence polarization competition binding assay using Plk. More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2012
Entry Details Article
PubMed