Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50039647
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 500nMAssay Description:Inhibition of mouse wild type PI3Kalpha expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 570nMAssay Description:Inhibition of PI3Kdelta expressed in cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol substrate by TLC based p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 970nMAssay Description:Inhibition of human wild type PI3Kbeta expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381605(CHEMBL2018409)
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of mouse wild type PI3Kalpha expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381603(CHEMBL2018266)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of PI3Kdelta expressed in cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol substrate by TLC based p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381605(CHEMBL2018409)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of human wild type PI3Kbeta expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381607(CHEMBL2018263)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of mouse wild type PI3Kalpha expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381604(CHEMBL2018271)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of mouse wild type PI3Kalpha expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381608(CHEMBL2018265)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of PI3Kdelta expressed in cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol substrate by TLC based p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381606(CHEMBL2018413)
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of PI3Kdelta expressed in cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol substrate by TLC based p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381604(CHEMBL2018271)
Affinity DataIC50: 2.97E+4nMAssay Description:Inhibition of PI3Kdelta expressed in cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol substrate by TLC based p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381603(CHEMBL2018266)
Affinity DataIC50: 3.12E+4nMAssay Description:Inhibition of mouse wild type PI3Kalpha expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381608(CHEMBL2018265)
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibition of mouse wild type PI3Kalpha expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381607(CHEMBL2018263)
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of human wild type PI3Kbeta expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381608(CHEMBL2018265)
Affinity DataIC50: 5.18E+4nMAssay Description:Inhibition of human wild type PI3Kbeta expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381606(CHEMBL2018413)
Affinity DataIC50: 5.49E+4nMAssay Description:Inhibition of mouse wild type PI3Kalpha expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381607(CHEMBL2018263)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PI3Kdelta expressed in cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol substrate by TLC based p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381606(CHEMBL2018413)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human wild type PI3Kbeta expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381604(CHEMBL2018271)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human wild type PI3Kbeta expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381605(CHEMBL2018409)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PI3Kdelta expressed in cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol substrate by TLC based p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50381603(CHEMBL2018266)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human wild type PI3Kbeta expressed in Sf21 cells co-expressing N-terminal His-tagged human p85a using L-alpha-phosphatidylinositol subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed