Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50041977
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420160(CHEMBL2058525)
Affinity DataEC50:  2.04E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275055(4-{4-[2-(Phenyl-2-pyridinylamino)ethoxy]phenyl}but...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22496(CHEMBL207881 | 3-(4-{[(3-phenoxyphenyl)methyl]amin...)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50240347((Z,Z,Z)-9,12,15-octadecatrienoic acid | cis,cis,ci...)
Affinity DataEC50:  3.24E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420165(CHEMBL2058531)
Affinity DataEC50:  407nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420164(CHEMBL2058530)
Affinity DataEC50:  110nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420148(CHEMBL2058529)
Affinity DataEC50:  603nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420163(CHEMBL2058528)
Affinity DataEC50:  3.55E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420162(CHEMBL2058527)
Affinity DataEC50:  631nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420161(CHEMBL2058526)
Affinity DataEC50:  4.47E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275597(3-(4-(o-Tolylethynyl)phenyl)propanoic acid | CHEMB...)
Affinity DataEC50:  2.24E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420159(CHEMBL2058524)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420158(CHEMBL2058523)
Affinity DataEC50:  851nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420157(CHEMBL2058522)
Affinity DataEC50:  513nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420156(CHEMBL2058521)
Affinity DataEC50:  933nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420155(CHEMBL2058520)
Affinity DataEC50:  631nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at FFAR1 expressed in Flp-In TREx293 cells by calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Mouse)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  17.0nMAssay Description:Agonist activity at mouse GPR120More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  95.5nMAssay Description:Agonist activity at GPR120 expressed in Flp-In TREx293 cells by calcium assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420171(CHEMBL1773255)
Affinity DataEC50:  741nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50339461(3-{4-[(3-Phenoxybenzyl)oxy]phenyl}propanoic Acid |...)
Affinity DataEC50:  562nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420166(CHEMBL2058532)
Affinity DataEC50:  955nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420167(CHEMBL2058533)
Affinity DataEC50:  6.46E+4nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420152(CHEMBL1773259)
Affinity DataEC50:  5.13E+4nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50339459(3-[4-(Biphenyl-2-ylmethoxy)phenyl]propanoic Acid |...)
Affinity DataEC50:  372nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420151(CHEMBL1773258)
Affinity DataEC50:  4.79E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50339460(3-[4-(Biphenyl-3-ylmethoxy)phenyl]propanoic Acid |...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22502(3-(4-{[(4-phenylphenyl)methyl]amino}phenyl)propano...)
Affinity DataEC50:  5.89E+4nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22528(3-(4-{[(4-phenoxyphenyl)methyl]amino}phenyl)propan...)
Affinity DataEC50:  4.47E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50339458(3-{4-[(4-Phenoxybenzyl)oxy]phenyl}propanoic Acid |...)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22510(3-(4-{[(3-bromophenyl)methyl]amino}phenyl)propanoi...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420150(CHEMBL1773256)
Affinity DataEC50:  6.76E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420149(CHEMBL1773257)
Affinity DataEC50:  1.29E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420171(CHEMBL1773255)
Affinity DataEC50:  2.09E+4nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22510(3-(4-{[(3-bromophenyl)methyl]amino}phenyl)propanoi...)
Affinity DataEC50:  3.09E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420170(CHEMBL1773254)
Affinity DataEC50:  479nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420169(CHEMBL1773253)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420168(CHEMBL1773252)
Affinity DataEC50:  5.37E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM22517(3-[4-(benzylamino)phenyl]propanoic acid | carboxyl...)
Affinity DataEC50:  5.75E+4nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50339456(Benzyloxyphenylpropanoic acid | CHEMBL1688452)
Affinity DataEC50:  1.17E+4nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420152(CHEMBL1773259)
Affinity DataEC50:  4.79E+3nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420155(CHEMBL2058520)
Affinity DataEC50:  178nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420154(CHEMBL2058519)
Affinity DataEC50:  1.95E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420153(CHEMBL2058518)
Affinity DataEC50:  7.08E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50343141(3-(4(2'-Methylbiphenyl-3-ylmethylamino)phenyl)prop...)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50339468(3-{4-[(2'-Methylbiphenyl-3-yl)methoxy]phenyl}propa...)
Affinity DataEC50:  8.71E+3nMAssay Description:Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420154(CHEMBL2058519)
Affinity DataEC50:  525nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50420153(CHEMBL2058518)
Affinity DataEC50:  603nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50343141(3-(4(2'-Methylbiphenyl-3-ylmethylamino)phenyl)prop...)
Affinity DataEC50:  12.9nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50339468(3-{4-[(2'-Methylbiphenyl-3-yl)methoxy]phenyl}propa...)
Affinity DataEC50:  16.6nMAssay Description:Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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