Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50045947
TargetSolute carrier family 15 member 1(Rat)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50088510(CHEMBL3526259)
Affinity DataKd:  2.20nMAssay Description:Activity at rat recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scintil...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Mouse)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50088510(CHEMBL3526259)
Affinity DataKd:  2.20nMAssay Description:Activity at mouse recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scint...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50088510(CHEMBL3526259)
Affinity DataKd:  2.20nMAssay Description:Activity at human recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scint...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Rat)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 1.83E+7nMAssay Description:Inhibition of rat recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation c...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Mouse)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 1.07E+7nMAssay Description:Inhibition of mouse recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM5025(ethyl (3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-y...)
Affinity DataIC50: 2.74E+7nMAssay Description:Inhibition of human recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as [3H]GlySar uptake after 30s by dual-channel liquid scintillation...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 6(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataKi:  4.51E+7nMAssay Description:Binding affinity to human OAT1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed