Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50039649
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381647(CHEMBL2023612)
Affinity DataKd:  0.0501nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381655(CHEMBL2021998)
Affinity DataKd:  0.0794nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381653(CHEMBL2021997)
Affinity DataKd:  0.0398nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381652(CHEMBL2023760)
Affinity DataKd:  0.0251nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381651(CHEMBL2023753)
Affinity DataKd:  0.158nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381650(CHEMBL2023752)
Affinity DataKd:  0.501nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381649(CHEMBL2023751)
Affinity DataKd:  1.26nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381648(CHEMBL2023750)
Affinity DataKd:  0.158nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381646(CHEMBL2023749)
Affinity DataKd:  0.0501nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381641(CHEMBL2023758)
Affinity DataKd:  0.631nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381640(CHEMBL2023613)
Affinity DataKd:  0.0501nMAssay Description:Antagonist potency at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381644(CHEMBL2023761)
Affinity DataIC50: 26.3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381645(CHEMBL2023763)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381643(CHEMBL2023759)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381642(CHEMBL2023757)
Affinity DataIC50: 85.2nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381637(CHEMBL2023754)
Affinity DataIC50: 89.6nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381639(CHEMBL2023756)
Affinity DataIC50: 109nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381638(CHEMBL2023755)
Affinity DataIC50: 318nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium mobilization b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381654(CHEMBL2023764)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]-N-methyl scopolamine from muscarinic acetylcholine M2 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381654(CHEMBL2023764)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]-N-methyl scopolamine from muscarinic acetylcholine M1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50381654(CHEMBL2023764)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-N-methyl scopolamine from muscarinic acetylcholine M3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed