Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50034666
TargetSodium channel protein type 9 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50365938(CHEMBL1958460)
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of human voltage-gated sodium channel 1.7 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50365939(CHEMBL1958461)
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of human voltage-gated sodium channel 1.7 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50365940(CHEMBL1958462)
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of human voltage-gated sodium channel 1.7 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50365940(CHEMBL1958462)
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of human voltage-gated sodium channel 1.5 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50365938(CHEMBL1958460)
Affinity DataIC50: 5.78E+3nMAssay Description:Inhibition of human voltage-gated sodium channel 1.5 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50365939(CHEMBL1958461)
Affinity DataIC50: 7.43E+3nMAssay Description:Inhibition of human voltage-gated sodium channel 1.5 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50003655(Phenytoin)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human voltage-gated sodium channel 1.5 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50003655(Phenytoin)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human voltage-gated sodium channel 1.7 expressed in HEK293 cells assessed as changes in membranre potential after 45 mins by FRET analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed