Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50004623
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289534(CHEMBL2018574)
Affinity DataEC50:  2.20E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50290134(CHEMBL2018580)
Affinity DataEC50:  4.20E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289860(CHEMBL2018582)
Affinity DataEC50:  6.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50290145(CHEMBL2018584)
Affinity DataEC50:  3.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289868(CHEMBL2018590)
Affinity DataEC50:  4.30E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289959(CHEMBL2018593)
Affinity DataEC50:  8.20E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289958(CHEMBL2018592)
Affinity DataEC50:  3.00E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM75164(N-[2-(3-Cyano-5,7-dimethyl-quinolin-2-ylamino)-eth...)
Affinity DataEC50:  1.10E+4nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50290130(CHEMBL2018575)
Affinity DataEC50:  3.00E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289859(CHEMBL2018581)
Affinity DataEC50:  1.50E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50290147(CHEMBL2018589)
Affinity DataEC50:  4.60E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50290144(CHEMBL2018578)
Affinity DataEC50:  7.30E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50290132(CHEMBL2018577)
Affinity DataEC50:  2.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289861(CHEMBL2018583)
Affinity DataEC50:  2.70E+3nMAssay Description:Activity at human CFTR delta F508 mutant expressed in forskolin-stimulated FRT cells assessed as increase in iodine influx measured as decrease in YF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed