Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50006063
TargetLysophosphatidic acid receptor 1/3(Rat)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50496697(CHEMBL3218460)
Affinity DataKi:  11nMAssay Description:Antagonist activity at LPAR1/LPAR3 in rat glioma C62B cells assessed as inhibition of LPA-induced reduction in isoproterenol-stimulated [3H]cAMP accu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50496698(CHEMBL3218459)
Affinity DataKi:  48nMAssay Description:Competitive antagonist activity at N-terminal 3XHA-tagged human LPA3 receptor overexpressed in CHO cells assessed as inhibition of LPA-induced [35S]G...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50496698(CHEMBL3218459)
Affinity DataKi:  84nMAssay Description:Competitive antagonist activity at human LPA1 receptor overexpressed in CHO cells assessed as inhibition of LPA-induced [35S]GTPgammaS binding by liq...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50496697(CHEMBL3218460)
Affinity DataKi:  143nMAssay Description:Competitive antagonist activity at human LPA1 receptor overexpressed in CHO cells assessed as inhibition of LPA-induced [35S]GTPgammaS binding by liq...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
University of Virginia

Curated by ChEMBL
LigandPNGBDBM50496697(CHEMBL3218460)
Affinity DataKi:  512nMAssay Description:Competitive antagonist activity at N-terminal 3XHA-tagged human LPA3 receptor overexpressed in CHO cells assessed as inhibition of LPA-induced [35S]G...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed