Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50034341
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50227631(2-(6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)iso...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360832(CHEMBL1934810)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360830(CHEMBL1934808)
Affinity DataIC50: 62nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360831(CHEMBL1934809)
Affinity DataIC50: 108nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360829(CHEMBL1934807)
Affinity DataIC50: 172nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360813(CHEMBL1934791)
Affinity DataIC50: 251nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360828(CHEMBL1934806)
Affinity DataIC50: 306nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360827(CHEMBL1934805)
Affinity DataIC50: 330nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360816(CHEMBL1934794)
Affinity DataIC50: 395nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360819(CHEMBL1934797)
Affinity DataIC50: 506nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360823(CHEMBL1934801)
Affinity DataIC50: 669nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360824(CHEMBL1934802)
Affinity DataIC50: 687nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360814(CHEMBL1934792)
Affinity DataIC50: 859nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360822(CHEMBL1934800)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360817(CHEMBL1934795)
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360826(CHEMBL1934804)
Affinity DataIC50: 4.12E+3nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360821(CHEMBL1934799)
Affinity DataIC50: 4.62E+3nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360825(CHEMBL1934803)
Affinity DataIC50: 6.26E+3nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360820(CHEMBL1934798)
Affinity DataIC50: 6.97E+3nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360812(CHEMBL1934678)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360818(CHEMBL1934796)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
Dainippon Sumitomo Pharma

Curated by ChEMBL
LigandPNGBDBM50360815(CHEMBL1934793)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of microsomal PGES1 transfected in human HEK293 cells assessed as PGE2 production after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed