Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50034335
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360737(CHEMBL1934473)
Affinity DataEC50: >6.80E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Dog)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  190nMAssay Description:Agonist activity at dog PPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360750(CHEMBL1934486)
Affinity DataEC50: >1.10E+4nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360749(CHEMBL1934485)
Affinity DataEC50:  1.80E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360748(CHEMBL1934484)
Affinity DataEC50:  3.10E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360747(CHEMBL1934483)
Affinity DataEC50:  8.80E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360746(CHEMBL1934482)
Affinity DataEC50:  1.90E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360745(CHEMBL1934481)
Affinity DataEC50:  2.40E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360744(CHEMBL1934480)
Affinity DataEC50:  7.10E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360743(CHEMBL1934479)
Affinity DataEC50: >1.30E+4nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Dog)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at dog PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360736(CHEMBL1934472)
Affinity DataEC50: >8.10E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360735(CHEMBL1934471)
Affinity DataEC50: >6.30E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360734(CHEMBL1934470)
Affinity DataEC50: >1.30E+4nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50: >4.20E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360754(CHEMBL1934314)
Affinity DataEC50: >1.70E+4nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360751(CHEMBL1934308)
Affinity DataEC50:  470nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50132472((S)-2-{3-[4-(4-Fluoro-phenoxy)-benzylcarbamoyl]-4-...)
Affinity DataEC50:  1.92E+3nMAssay Description:Transactivation of human PPARdelta expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360750(CHEMBL1934486)
Affinity DataEC50: >1.30E+4nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360756(CHEMBL1934309)
Affinity DataEC50:  4.40E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360755(CHEMBL1934468)
Affinity DataEC50:  280nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  5nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360760(CHEMBL1934316)
Affinity DataEC50: >1.20E+4nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360759(CHEMBL1934315)
Affinity DataEC50: >1.40E+4nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360754(CHEMBL1934314)
Affinity DataEC50:  810nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360758(CHEMBL1934313)
Affinity DataEC50:  700nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360753(CHEMBL1934312)
Affinity DataEC50:  850nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360757(CHEMBL1934311)
Affinity DataEC50: >3.50E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360752(CHEMBL1934310)
Affinity DataEC50:  760nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360749(CHEMBL1934485)
Affinity DataEC50: >1.10E+4nMAssay Description:Transactivation of human PPARgamma expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360751(CHEMBL1934308)
Affinity DataEC50:  700nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50132472((S)-2-{3-[4-(4-Fluoro-phenoxy)-benzylcarbamoyl]-4-...)
Affinity DataEC50:  13nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Mouse)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Mouse)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at mouse PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at mouse PPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at rat PPARgammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Rat)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at rat PPARalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Dog)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360740(CHEMBL1934476)
Affinity DataEC50:  2.70E+3nMAssay Description:Agonist activity at dog PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360739(CHEMBL1934475)
Affinity DataEC50:  1.50E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360749(CHEMBL1934485)
Affinity DataEC50:  23nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360748(CHEMBL1934484)
Affinity DataEC50:  6nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360747(CHEMBL1934483)
Affinity DataEC50:  21nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360746(CHEMBL1934482)
Affinity DataEC50:  53nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360745(CHEMBL1934481)
Affinity DataEC50:  26nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360744(CHEMBL1934480)
Affinity DataEC50:  72nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360743(CHEMBL1934479)
Affinity DataEC50:  1.50E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360742(CHEMBL1934478)
Affinity DataEC50: >3.40E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360741(CHEMBL1934477)
Affinity DataEC50:  1.20E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360750(CHEMBL1934486)
Affinity DataEC50:  37nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50360738(CHEMBL1934474)
Affinity DataEC50: >6.00E+3nMAssay Description:Transactivation of human PPARalpha expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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