Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50034314
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360416(CHEMBL1934260)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360419(CHEMBL1934253)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360418(CHEMBL1934264)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360420(CHEMBL1934254)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360418(CHEMBL1934264)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360416(CHEMBL1934260)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360417(CHEMBL1934265)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360422(CHEMBL1934256)
Affinity DataIC50: 78nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360421(CHEMBL1934259)
Affinity DataIC50: 98nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360419(CHEMBL1934253)
Affinity DataIC50: 98nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50355069(CHEMBL1835756)
Affinity DataIC50: 112nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360421(CHEMBL1934259)
Affinity DataIC50: 122nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360417(CHEMBL1934265)
Affinity DataIC50: 139nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360424(CHEMBL1934255)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360415(CHEMBL1934263)
Affinity DataIC50: 186nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360423(CHEMBL1934258)
Affinity DataIC50: 188nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360420(CHEMBL1934254)
Affinity DataIC50: 248nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360414(CHEMBL1934262)
Affinity DataIC50: 264nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360424(CHEMBL1934255)
Affinity DataIC50: 279nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360422(CHEMBL1934256)
Affinity DataIC50: 393nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50355069(CHEMBL1835756)
Affinity DataIC50: 476nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360425(CHEMBL1934257)
Affinity DataIC50: 799nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360425(CHEMBL1934257)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360423(CHEMBL1934258)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360414(CHEMBL1934262)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataIC50: 3.41E+3nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360413(CHEMBL1934261)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360415(CHEMBL1934263)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360413(CHEMBL1934261)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at human B1 bradykinin receptor expressed in CHO cells by aqueorin-based calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Rabbit)
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataIC50: 6.47E+3nMAssay Description:Antagonist activity at rabbit B1 bradykinin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360416(CHEMBL1934260)
Affinity DataKi:  4nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360417(CHEMBL1934265)
Affinity DataKi:  15nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360418(CHEMBL1934264)
Affinity DataKi:  17nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360420(CHEMBL1934254)
Affinity DataKi:  29nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360414(CHEMBL1934262)
Affinity DataKi:  42nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360419(CHEMBL1934253)
Affinity DataKi:  43nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50355069(CHEMBL1835756)
Affinity DataKi:  64nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360421(CHEMBL1934259)
Affinity DataKi:  184nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360423(CHEMBL1934258)
Affinity DataKi:  322nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360422(CHEMBL1934256)
Affinity DataKi:  398nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360415(CHEMBL1934263)
Affinity DataKi:  481nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360424(CHEMBL1934255)
Affinity DataKi:  767nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50360413(CHEMBL1934261)
Affinity DataKi:  1.62E+3nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetB1 bradykinin receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50355083(CHEMBL1835762)
Affinity DataKi:  6.37E+3nMAssay Description:Binding affinity to human B1 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed