Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50034394
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361658(CHEMBL1940482)
Affinity DataIC50: 17nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361660(CHEMBL1940599)
Affinity DataIC50: 22nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361654(CHEMBL1940477)
Affinity DataIC50: 324nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361659(CHEMBL1940597)
Affinity DataIC50: 1.99E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361656(CHEMBL1940479)
Affinity DataIC50: 2.91E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361655(CHEMBL1940478)
Affinity DataIC50: 6.64E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rat)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361657(CHEMBL1940480)
Affinity DataIC50: 7.14E+3nMAssay Description:Displacement of [3H]ifenprodil from GluN2B/NMDA in Wistar rat cerebral cortex after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361661(CHEMBL1940484)
Affinity DataKi:  437nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50276978(1-(4-benzylpiperidin-1-yl)-2-(5-hydroxy-1Hindol-3-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361660(CHEMBL1940599)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50361658(CHEMBL1940482)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
University of Messina

Curated by ChEMBL
LigandPNGBDBM50276976(2-(4-benzylpiperidin-1-yl)-1-(5-hydroxy-1Hindol-3-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H](+)pentazocine from sigma 1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed