Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 5656
TargetMyeloperoxidase(Human)
Astrazeneca R&D

LigandPNGBDBM92467(2-Thioxanthine, TX2)
Affinity DataIC50: 200nMpH: 7.4 T: 2°CAssay Description:The chlorination activity of MPO was determined by measuring the production of hypocholorous acid. More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMyeloperoxidase(Human)
Astrazeneca R&D

LigandPNGBDBM92469(2-Thioxanthine, TX4)
Affinity DataIC50: 200nMpH: 7.4 T: 2°CAssay Description:The chlorination activity of MPO was determined by measuring the production of hypocholorous acid. More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed
TargetMyeloperoxidase(Human)
Astrazeneca R&D

LigandPNGBDBM92468(2-Thioxanthine, TX3)
Affinity DataIC50: 400nMpH: 7.4 T: 2°CAssay Description:The chlorination activity of MPO was determined by measuring the production of hypocholorous acid. More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed
TargetMyeloperoxidase(Human)
Astrazeneca R&D

LigandPNGBDBM92470(2-Thioxanthine, TX5)
Affinity DataIC50: 400nMpH: 7.4 T: 2°CAssay Description:The chlorination activity of MPO was determined by measuring the production of hypocholorous acid. More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMyeloperoxidase(Human)
Astrazeneca R&D

LigandPNGBDBM92466(2-Thioxanthine, TX1)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:The chlorination activity of MPO was determined by measuring the production of hypocholorous acid. More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2012
Entry Details Article
PubMed