Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50004559
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM1434(BI-RG-587 | 2-cyclopropyl-7-methyl-2,4,9,15-tetraa...)
Affinity DataIC50: 670nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2184(SM30 | US8501787, 166)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2173(CW23836 | US8501787, 116)
Affinity DataIC50: 3.47E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2172(DG 402-49748 | US8501787, 104)
Affinity DataIC50: 3.74E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2115(MLB133-641A | US8501787, 8)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2116(DG 402-49706 | US8501787, 42)
Affinity DataIC50: 4.62E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2177(SM27 | US8501787, 163)
Affinity DataIC50: 5.39E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM99893(US8501767, 96)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2182(SM29 | US8501787, 165)
Affinity DataIC50: 7.18E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM2162(DG 402-49754 | US8501787, 97)
Affinity DataIC50: 7.52E+3nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM99895(US8501767, 81)
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM99896(US8501767, 99)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM99894(US8501767, 82)
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Csir Biosciences

Curated by ChEMBL
LigandPNGBDBM50484067(CHEMBL1807349)
Affinity DataIC50: 1.89E+4nMAssay Description:Inhibition of HIV1 reverse transcriptase assessed as residual enzyme activity at 50 uM after 1 hr by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed