Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50004548
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50483961(CHEMBL1795561)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human recombinant GABA A receptor alpha1beta2gamma2S expressed in HEK293 cells assessed as inhibition of GABA-induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50483959(CHEMBL1795560)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human recombinant GABA A receptor alpha1beta2gamma2S expressed in HEK293 cells assessed as inhibition of GABA-induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50483958(CHEMBL1795348)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human recombinant GABA A receptor alpha1beta2gamma2S expressed in HEK293 cells assessed as inhibition of GABA-induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50483960(CHEMBL1795562)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human recombinant GABA A receptor alpha1beta2gamma2S expressed in HEK293 cells assessed as inhibition of GABA-induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50001572(4-(6-imino-3-(4-methoxyphenyl)pyridazin-1(6H)-yl)b...)
Affinity DataIC50: 349nMAssay Description:Antagonist activity at human recombinant GABA A receptor alpha1beta2gamma2S expressed in HEK293 cells assessed as inhibition of GABA-induced current ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed