Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50048826
LigandPNGBDBM82427(CAS_5985-38-6 | LEVORPHANOL-tartarate)
Affinity DataIC50: 4.80nMAssay Description:Concentration that produces 50% inhibition of stereospecific [3H]naloxone binding to opioid receptors in rat brain in absence of sodium.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2019
Entry Details Article
PubMed
LigandPNGBDBM82427(CAS_5985-38-6 | LEVORPHANOL-tartarate)
Affinity DataIC50: 57nMAssay Description:Concentration that produces 50% inhibition of stereospecific [3H]naloxone binding to opioid receptors in rat brain in presence of sodium.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2019
Entry Details Article
PubMed
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataIC50: 226nMAssay Description:Concentration that produces 50% inhibition of stereospecific [3H]naloxone binding to opioid receptors in rat brain in absence of sodium.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2019
Entry Details Article
PubMed
LigandPNGBDBM50228352(CHEMBL81058)
Affinity DataIC50: 472nMAssay Description:Concentration that produces 50% inhibition of stereospecific [3H]naloxone binding to opioid receptors in rat brain in absence of sodium.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2019
Entry Details Article
PubMed
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataIC50: 487nMAssay Description:Concentration that produces 50% inhibition of stereospecific [3H]naloxone binding to opioid receptors in rat brain in presence of sodium.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2019
Entry Details Article
PubMed
LigandPNGBDBM50228352(CHEMBL81058)
Affinity DataIC50: 5.59E+3nMAssay Description:Concentration that produces 50% inhibition of stereospecific [3H]naloxone binding to opioid receptors in rat brain in presence of sodium.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/12/2019
Entry Details Article
PubMed