Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50033332
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343452(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50:  15.5nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343451(isobutyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazo...)
Affinity DataEC50:  4.20nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343452(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50:  5.60nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343453(tert-butyl 4-((ethyl(1-(4-(methylsulfonyl)phenyl)-...)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343434(tert-butyl 4-((1-(4-(methylsulfonyl)phenyl)-1H-pyr...)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343443(tert-butyl 4-(1-(2-fluoro-4-(methylsulfonyl)phenyl...)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343454(tert-butyl 4-(3-(4-(methylsulfonyl)phenyl)-3H-[1,2...)
Affinity DataEC50:  7.40nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343455(butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[...)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343456(neopentyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyraz...)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343447(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50:  9.80nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343457(tert-butyl 4-((methyl(1-(4-(methylsulfonyl)phenyl)...)
Affinity DataEC50:  11.6nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343458(isopropyl 4-(3-(4-(methylsulfonyl)phenyl)isoxazolo...)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343459(cyclopentyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyr...)
Affinity DataEC50:  14.6nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343460(tert-butyl 4-(3-methyl-1-(4-(methylsulfonyl)phenyl...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343450(ethyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[...)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343445(tert-butyl 4-(3-(4-(methylsulfonyl)phenyl)isoxazol...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343446(tert-butyl 4-(1-(2-fluoro-4-(methylsulfonyl)phenyl...)
Affinity DataEC50:  19.6nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343459(cyclopentyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyr...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343442(isopropyl 4-(1-(2-fluoro-4-(methylsulfonyl)phenyl)...)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human GPR119 expressed in human HEK293 cells assessed as increase in adenylate cyclase activationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343442(isopropyl 4-(1-(2-fluoro-4-(methylsulfonyl)phenyl)...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343461(tert-butyl 4-(9-(4-(methylsulfonyl)phenyl)-9H-puri...)
Affinity DataEC50:  33.4nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343458(isopropyl 4-(3-(4-(methylsulfonyl)phenyl)isoxazolo...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343460(tert-butyl 4-(3-methyl-1-(4-(methylsulfonyl)phenyl...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343454(tert-butyl 4-(3-(4-(methylsulfonyl)phenyl)-3H-[1,2...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343450(ethyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[...)
Affinity DataEC50:  53nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343456(neopentyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyraz...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343448(tert-butyl 4-((1-(2-fluoro-4-(methylsulfonyl)pheny...)
Affinity DataEC50:  88nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343439(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50244680({6-[4-(3-Isopropyl-[1,2,4]oxadiazol-5-yl)-piperidi...)
Affinity DataEC50:  5.10nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50244791((2-Fluoro-4-methanesulfonyl-phenyl)-{6-[4-(3-isopr...)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343433(tert-butyl 4-(3,6-dimethyl-1-(4-(methylsulfonyl)ph...)
Affinity DataEC50:  116nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343434(tert-butyl 4-((1-(4-(methylsulfonyl)phenyl)-1H-pyr...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343435(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343436(isopropyl 4-((ethyl(1-(2-fluoro-4-(methylsulfonyl)...)
Affinity DataEC50:  264nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343437(tert-butyl 4-((1-(4-(methylsulfonyl)phenyl)-1H-pyr...)
Affinity DataEC50:  265nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343438(tetrahydrofuran-3-yl 4-(1-(4-(methylsulfonyl)pheny...)
Affinity DataEC50:  435nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343439(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343440(2-(dimethylamino)ethyl 4-(1-(4-(methylsulfonyl)phe...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343441(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343435(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343432(3-isopropyl-5-(1-(1-(4-(methylsulfonyl)phenyl)-1H-...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Rat)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343441(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343443(tert-butyl 4-(1-(2-fluoro-4-(methylsulfonyl)phenyl...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343444(tert-butyl 4-(9-(2-fluoro-4-(methylsulfonyl)phenyl...)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343445(tert-butyl 4-(3-(4-(methylsulfonyl)phenyl)isoxazol...)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343446(tert-butyl 4-(1-(2-fluoro-4-(methylsulfonyl)phenyl...)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343447(tert-butyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyra...)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343442(isopropyl 4-(1-(2-fluoro-4-(methylsulfonyl)phenyl)...)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343436(isopropyl 4-((ethyl(1-(2-fluoro-4-(methylsulfonyl)...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50343448(tert-butyl 4-((1-(2-fluoro-4-(methylsulfonyl)pheny...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human GPR119 by melanophore assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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