Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50033134
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340102(N-ethyl-N-(3-fluoropropyl)-8-(6-methoxy-2-methylpy...)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340103(N-(3-fluoropropyl)-8-(6-methoxy-2-methylpyridin-3-...)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340101(N-(2-fluoroethyl)-8-(6-methoxy-2-methylpyridin-3-y...)
Affinity DataIC50: 5.5nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340100(N-ethyl-N-(2-fluoroethyl)-8-(6-methoxy-2-methylpyr...)
Affinity DataIC50: 5.80nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340104(3-((3-fluoropropyl)(8-(6-methoxy-2-methylpyridin-3...)
Affinity DataIC50: 6.5nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340105(N-(3-fluoropropyl)-N-(2-methoxyethyl)-8-(6-methoxy...)
Affinity DataIC50: 35nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340106(N-(3-fluoropropyl)-N-(2-methoxyethyl)-8-(2-methoxy...)
Affinity DataIC50: 390nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50340107(8-(2,4-dimethoxypyrimidin-5-yl)-N-(3-fluoropropyl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-o-CRF from CRF1 receptor in rat frontal cortex by rapid filtration techniqueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed