Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50001117
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataIC50: 680nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(CHEMBL339944 | 3-(3-Piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(CHEMBL339944 | 3-(3-Piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(CHEMBL339944 | 3-(3-Piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(CHEMBL339944 | 3-(3-Piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(CHEMBL341326 | 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(CHEMBL341326 | 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(CHEMBL128329 | 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(CHEMBL128329 | 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(CHEMBL128329 | 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl...)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(CHEMBL128329 | 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl...)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(CHEMBL341326 | 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(CHEMBL341326 | 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(CHEMBL128954 | 5-Phenyl-6-piperidin-1-yl-bicyclo[2...)
Affinity DataIC50: 1.81E+5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(CHEMBL128954 | 5-Phenyl-6-piperidin-1-yl-bicyclo[2...)
Affinity DataIC50: 3.58E+5nMAssay Description:Inhibitory activity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  500nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(CHEMBL339944 | 3-(3-Piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataKi:  8.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(CHEMBL339944 | 3-(3-Piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataKi:  8.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(CHEMBL341326 | 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataKi:  8.50E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012983(CHEMBL339944 | 3-(3-Piperidin-1-yl-bicyclo[2.2.2]o...)
Affinity DataKi:  1.35E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(CHEMBL341326 | 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataKi:  1.70E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012982(CHEMBL341326 | 3-(3-Pyrrolidin-1-yl-bicyclo[2.2.2]...)
Affinity DataKi:  1.70E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(CHEMBL128329 | 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl...)
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(CHEMBL128329 | 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl...)
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012980(CHEMBL128329 | 5-(1H-Indol-3-yl)-6-pyrrolidin-1-yl...)
Affinity DataKi:  3.20E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataKi:  6.10E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012981(CHEMBL338310 | 5-(1H-Indol-3-yl)-6-piperidin-1-yl-...)
Affinity DataKi:  6.10E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A/2B/2C(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(CHEMBL128954 | 5-Phenyl-6-piperidin-1-yl-bicyclo[2...)
Affinity DataKi:  1.32E+5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptor by the displacement of [3H]-ketanserin in mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
Polytechnic University

Curated by ChEMBL
LigandPNGBDBM50012984(CHEMBL128954 | 5-Phenyl-6-piperidin-1-yl-bicyclo[2...)
Affinity DataKi:  2.74E+5nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor by the displacement of [3H]8-OH-DPAT in mouse hippocampusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed