Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50033322
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343293(6-[5-(Cyclopropylmethyl)-4,5-dihydro-1'H,3H-spiro[...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343293(6-[5-(Cyclopropylmethyl)-4,5-dihydro-1'H,3H-spiro[...)
Affinity DataIC50: 10nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343291(N-(2-Hydroxy-2-pyridin-3-ylethyl)-6-(5-isopropyl-4...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343291(N-(2-Hydroxy-2-pyridin-3-ylethyl)-6-(5-isopropyl-4...)
Affinity DataIC50: 40nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343290(6-(5-Ethyl-4,5-dihydro-1'H,3H-spiro[1,5-benzoxazep...)
Affinity DataIC50: 40nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50306110(N-(2-hydroxy-2-phenylethyl)-6-(4-oxospiro[chroman-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343288(N-(2-hydroxy-2-phenylethyl)-6-(5-methyl-4,5-dihydr...)
Affinity DataIC50: 50nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343290(6-(5-Ethyl-4,5-dihydro-1'H,3H-spiro[1,5-benzoxazep...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50306110(N-(2-hydroxy-2-phenylethyl)-6-(4-oxospiro[chroman-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343288(N-(2-hydroxy-2-phenylethyl)-6-(5-methyl-4,5-dihydr...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343289(N-(2-Hydroxy-2-pyridin-3-ylethyl)-6-(5-methyl-4,5-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343294(6-[5-(2-Hydroxyethyl)-4,5-dihydro-1'H,3H-spiro[1,5...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343289(N-(2-Hydroxy-2-pyridin-3-ylethyl)-6-(5-methyl-4,5-...)
Affinity DataIC50: 700nMAssay Description:Inhibition of human SCD1 transfected in human 293A cells after 30 mins by whole cell assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343287(6-(4,5-dihydro-3H-spiro[benzo[b][1,4]oxazepine-2,4...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343287(6-(4,5-dihydro-3H-spiro[benzo[b][1,4]oxazepine-2,4...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343286(N-(2-hydroxy-2-phenylethyl)-6-(4-oxo-4,5-dihydro-3...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343286(N-(2-hydroxy-2-phenylethyl)-6-(4-oxo-4,5-dihydro-3...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetStearoyl-CoA desaturase(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343285(N-(2-hydroxy-2-(pyridin-3-yl)ethyl)-6-(4-oxospiro[...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343294(6-[5-(2-Hydroxyethyl)-4,5-dihydro-1'H,3H-spiro[1,5...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAcyl-CoA desaturase 1(Mouse)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50343292(6-(5-Cyclopropyl-4,5-dihydro-1'H,3H-spiro[1,5-benz...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of mouse liver microsome SCD1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed