Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 5650
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM7918(PBD150 | 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dim...)
Affinity DataKi:  95nM ΔG°:  -40.1kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM7887(1-benzylimidazole | 1-Benzylimidazole (BI) | CHEMB...)
Affinity DataKi:  262nM ΔG°:  -37.6kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM7887(1-benzylimidazole | 1-Benzylimidazole (BI) | CHEMB...)
Affinity DataKi:  607nM ΔG°:  -35.5kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM7949(N-[2-(1H-Imidazol-4-yl)ethyl]acetamide | N-omega-A...)
Affinity DataKi:  1.70E+3nM ΔG°:  -32.9kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM7918(PBD150 | 1-(3-(1H-Imidazol-1-yl)propyl)-3-(3,4-dim...)
Affinity DataKi:  1.82E+3nM ΔG°:  -32.8kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM7949(N-[2-(1H-Imidazol-4-yl)ethyl]acetamide | N-omega-A...)
Affinity DataKi:  5.75E+3nM ΔG°:  -29.9kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM92451(Cacodylate)
Affinity DataKi:  6.70E+6nM ΔG°:  -12.4kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Academia Sinica

LigandPNGBDBM92451(Cacodylate)
Affinity DataKi:  1.82E+6nM ΔG°:  -15.6kJ/molepH: 8.0 T: 2°CAssay Description:The testing for the inhibition activities of imidazole derivatives and cacodylate on gQC and sQC was evaluated at 25 C using the fluorescent substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/10/2012
Entry Details Article
PubMed