Compile Data Set for Download or QSAR
Report error Found 131 Enz. Inhib. hit(s) with all data for entry = 50032983
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337366(2-(1H-indazol-5-yl)-3-phenylimidazo[1,2-a]pyrimidi...)
Affinity DataKi:  6nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337385(5-(1-(1-benzylpyrrolidin-3-yl)-4-(4-fluorophenyl)-...)
Affinity DataKi:  8nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337366(2-(1H-indazol-5-yl)-3-phenylimidazo[1,2-a]pyrimidi...)
Affinity DataKi:  10nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337377(N-cyclohexyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyri...)
Affinity DataKi:  10nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337383(4-(2-(4-(4-fluorophenyl)-5-(1H-indazol-5-yl)-1H-im...)
Affinity DataKi:  17nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337378(2-(1H-indazol-5-yl)-N-isopropylimidazo[1,2-a]pyrim...)
Affinity DataKi:  17nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337379(N-butyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyrimidin...)
Affinity DataKi:  19nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337384(4-(3-(4-(4-fluorophenyl)-5-(1H-indazol-5-yl)-1H-im...)
Affinity DataKi:  27nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337378(2-(1H-indazol-5-yl)-N-isopropylimidazo[1,2-a]pyrim...)
Affinity DataKi:  65nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337382(2-(4-(4-fluorophenyl)-5-(1H-indazol-5-yl)-1H-imida...)
Affinity DataKi:  67nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337379(N-butyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyrimidin...)
Affinity DataKi:  114nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337379(N-butyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyrimidin...)
Affinity DataKi:  116nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337380(N-(4-chlorophenyl)-2-(1H-indazol-5-yl)imidazo[1,2-...)
Affinity DataKi:  121nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337371(N-benzyl-4-(1H-indazol-5-yl)thiazol-2-amine | CHEM...)
Affinity DataKi:  136nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337365(2-(1H-indazol-5-yl)imidazo[1,2-a]pyrimidine | CHEM...)
Affinity DataKi:  141nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337365(2-(1H-indazol-5-yl)imidazo[1,2-a]pyrimidine | CHEM...)
Affinity DataKi:  226nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337378(2-(1H-indazol-5-yl)-N-isopropylimidazo[1,2-a]pyrim...)
Affinity DataKi:  242nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337377(N-cyclohexyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyri...)
Affinity DataKi:  245nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337370(4-(1H-indazol-5-yl)-N-phenylthiazol-2-amine | CHEM...)
Affinity DataKi:  289nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337377(N-cyclohexyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyri...)
Affinity DataKi:  307nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337366(2-(1H-indazol-5-yl)-3-phenylimidazo[1,2-a]pyrimidi...)
Affinity DataKi:  339nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337372(4-(1H-indazol-5-yl)-N-phenethylthiazol-2-amine | C...)
Affinity DataKi:  364nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337367(4-(1H-indazol-5-yl)-2-methylthiazole | CHEMBL16825...)
Affinity DataKi:  513nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAurora kinase B(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337371(N-benzyl-4-(1H-indazol-5-yl)thiazol-2-amine | CHEM...)
Affinity DataKi:  588nMAssay Description:Inhibition of aurora 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337381(N-cyclohexyl-6-(1H-indazol-5-yl)imidazo[2,1-b]thia...)
Affinity DataKi:  622nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337381(N-cyclohexyl-6-(1H-indazol-5-yl)imidazo[2,1-b]thia...)
Affinity DataKi:  642nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAurora kinase B(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337372(4-(1H-indazol-5-yl)-N-phenethylthiazol-2-amine | C...)
Affinity DataKi:  810nMAssay Description:Inhibition of aurora 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337374(N-benzyl-4-(1H-indazol-5-yl)-5-phenylthiazol-2-ami...)
Affinity DataKi:  822nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAurora kinase B(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337370(4-(1H-indazol-5-yl)-N-phenylthiazol-2-amine | CHEM...)
Affinity DataKi:  834nMAssay Description:Inhibition of aurora 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337370(4-(1H-indazol-5-yl)-N-phenylthiazol-2-amine | CHEM...)
Affinity DataKi:  864nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337369(N-ethyl-4-(1H-indazol-5-yl)thiazol-2-amine | CHEMB...)
Affinity DataKi:  888nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337368(4-(1H-indazol-5-yl)thiazol-2-amine | CHEMBL1682543)
Affinity DataKi:  909nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337381(N-cyclohexyl-6-(1H-indazol-5-yl)imidazo[2,1-b]thia...)
Affinity DataKi:  1.29E+3nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337373(4-(1H-indazol-5-yl)-N,5-diphenylthiazol-2-amine | ...)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337371(N-benzyl-4-(1H-indazol-5-yl)thiazol-2-amine | CHEM...)
Affinity DataKi: >1.45E+3nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337382(2-(4-(4-fluorophenyl)-5-(1H-indazol-5-yl)-1H-imida...)
Affinity DataKi: >1.45E+3nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337383(4-(2-(4-(4-fluorophenyl)-5-(1H-indazol-5-yl)-1H-im...)
Affinity DataKi: >1.45E+3nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337384(4-(3-(4-(4-fluorophenyl)-5-(1H-indazol-5-yl)-1H-im...)
Affinity DataKi: >1.45E+3nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337385(5-(1-(1-benzylpyrrolidin-3-yl)-4-(4-fluorophenyl)-...)
Affinity DataKi: >1.45E+3nMAssay Description:Inhibition of JAK2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRho-associated protein kinase 2(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337380(N-(4-chlorophenyl)-2-(1H-indazol-5-yl)imidazo[1,2-...)
Affinity DataKi:  1.57E+3nMAssay Description:Inhibition of Rock2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337365(2-(1H-indazol-5-yl)imidazo[1,2-a]pyrimidine | CHEM...)
Affinity DataKi:  1.66E+3nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337365(2-(1H-indazol-5-yl)imidazo[1,2-a]pyrimidine | CHEM...)
Affinity DataKi: >1.80E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337370(4-(1H-indazol-5-yl)-N-phenylthiazol-2-amine | CHEM...)
Affinity DataKi: >1.80E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337371(N-benzyl-4-(1H-indazol-5-yl)thiazol-2-amine | CHEM...)
Affinity DataKi: >1.80E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337377(N-cyclohexyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyri...)
Affinity DataKi: >1.80E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEpidermal growth factor receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337378(2-(1H-indazol-5-yl)-N-isopropylimidazo[1,2-a]pyrim...)
Affinity DataKi: >1.80E+3nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337376(N-cyclohexyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyra...)
Affinity DataKi:  1.85E+3nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337369(N-ethyl-4-(1H-indazol-5-yl)thiazol-2-amine | CHEMB...)
Affinity DataKi:  1.95E+3nMAssay Description:Inhibition of Pim1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAurora kinase B(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337376(N-cyclohexyl-2-(1H-indazol-5-yl)imidazo[1,2-a]pyra...)
Affinity DataKi:  2.07E+3nMAssay Description:Inhibition of aurora 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAurora kinase B(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50337368(4-(1H-indazol-5-yl)thiazol-2-amine | CHEMBL1682543)
Affinity DataKi:  2.13E+3nMAssay Description:Inhibition of aurora 2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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