Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50032650
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  15nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332720((S)-1-((4R,7S,10S,13S,16S,19R)-4-amino-16-(2-amino...)
Affinity DataEC50:  2.60nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332730((R)-N-((R)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataEC50: >1.00E+5nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332729((4S,7R,10S,13R,16R,19S)-16-(2-amino-2-oxoethyl)-13...)
Affinity DataEC50: >1.00E+5nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332728(cyclo(CYIQNCPLGAGAGAG | CHEMBL1630533)
Affinity DataEC50: >1.00E+5nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332725((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataEC50:  18nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332724((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataEC50:  27.3nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332723(Cystathionine Oxytocin | CHEMBL1630531)
Affinity DataEC50:  32nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50291330(AVP (Arginine-vasopressin ) | 1-[19-Amino-13-benzy...)
Affinity DataEC50:  41nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332721((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataEC50:  154nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332727(cyclo(CYIQNCPLG) | CHEMBL1630532)
Affinity DataEC50: >1.00E+5nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332726(Lanthionine Oxytocin | CHEMBL1630530)
Affinity DataEC50: >1.00E+5nMAssay Description:Activity at oxytocin receptor expressed in COS1 cells assessed as IP-one generation by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332720((S)-1-((4R,7S,10S,13S,16S,19R)-4-amino-16-(2-amino...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332721((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.790nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332723(Cystathionine Oxytocin | CHEMBL1630531)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332724((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332725((S)-N-((S)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataKi:  11.8nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50291330(AVP (Arginine-vasopressin ) | 1-[19-Amino-13-benzy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332726(Lanthionine Oxytocin | CHEMBL1630530)
Affinity DataKi:  856nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332727(cyclo(CYIQNCPLG) | CHEMBL1630532)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332726(Lanthionine Oxytocin | CHEMBL1630530)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332728(cyclo(CYIQNCPLGAGAGAG | CHEMBL1630533)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332729((4S,7R,10S,13R,16R,19S)-16-(2-amino-2-oxoethyl)-13...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetOxytocin receptor(Human)
The University of Queensland

Curated by ChEMBL
LigandPNGBDBM50332730((R)-N-((R)-1-(2-amino-2-oxoethylamino)-3-methylbut...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]OT from oxytocin receptor expressed in COS1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed