Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50032625
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM17762(3-[2-carboxy-2-(3-sulfanylpropyl)ethyl]benzoic aci...)
Affinity DataIC50: 15nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332217(1-[(2-carboxyphenyl)methyl]-3-(2-mercaptoethyl)-1H...)
Affinity DataIC50: 22nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332218(1-[(3-carboxyphenyl)methyl]-3-(2-mercaptoethyl)-1H...)
Affinity DataIC50: 22nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332228(1-(3-Carboxyphenyl)-3-(2-mercapto-ethyl)-1H-indole...)
Affinity DataIC50: 22nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332221(1-[[3-carboxy-5-(1,1-dimethylethyl)phenyl]methyl]-...)
Affinity DataIC50: 34nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332220(1-[(2-bromo-5-carboxyphenyl)methyl]-3-(2-mercaptoe...)
Affinity DataIC50: 54nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM17755(pentanedioic acid analogue, (RS)-3 | CHEMBL303352 ...)
Affinity DataIC50: 90nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332223(1-[(2-carboxy-5-methoxyphenyl)methyl]-3-(2-mercapt...)
Affinity DataIC50: 93nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332219(1-[(4-carboxyphenyl)methyl]-3-(2-mercaptoethyl)-1H...)
Affinity DataIC50: 94nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332222(1-[(4-bromo-3-carboxyphenyl)methyl]-3-(2-mercaptoe...)
Affinity DataIC50: 140nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332215(3-(2-Mercaptoethyl)-1H-indole-2-carboxylic acid | ...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332226(1-(3-Carboxybenzyl)-3-(carboxymethyl)-1H-indole-2-...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332227(3-(2-mercaptoethyl)-1-phenyl-1H-indole-2-carboxyli...)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332216(3-(2-Mercaptoethyl)-1-(phenylmethyl)-1H-indole-2-c...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332225(1-[(3-carboxyphenyl)methyl]-3-(2-methylsulfanyleth...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50332224(1-(3-carboxybenzyl)-3-(2-hydroxyethyl)-1H-indole-2...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Eisai Research Institute

Curated by ChEMBL
LigandPNGBDBM50246899(N-{[(1S)-1-carboxy-5-{[(4-iodophenyl)carbonyl]amin...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of GCP2 by top scintillation counter in presence of 30 nM NAA[3]GMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed