Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50032384
LigandPNGBDBM50328264(5-(2-chlorophenyl)-3-isopropyl-7-nitro-2,10-dihydr...)
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328256(5-(2-fluorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 16nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328279(5-(2-fluorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 17nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328267(5-(2-chlorophenyl)-7-nitro-3-(1H-pyrrol-2-yl)-2,10...)
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328280(N-(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo...)
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328258(N-(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo...)
Affinity DataIC50: 33nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328257(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 34nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328255(5-(2-chlorophenyl)-3-methyl-7-nitro-2,10-dihydrobe...)
Affinity DataIC50: 35nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328258(N-(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo...)
Affinity DataIC50: 38nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328256(5-(2-fluorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 39nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328274(7-fluoro-5-(2-fluorophenyl)-3-methyl-2,10-dihydrob...)
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328281(N'-[5-(2-chlorophenyl)-2,10-dihydropyrazolo[3,4-b]...)
Affinity DataIC50: 46nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328269(5-(2-chlorophenyl)-7-nitro-3-(pyridin-4-yl)-2,10-d...)
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328272(5-(2-fluorophenyl)-3-methyl-2,10-dihydrobenzo[e]py...)
Affinity DataIC50: 64nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328260(5-(2-chlorophenyl)-7-nitro-2,10-dihydrobenzo[e]pyr...)
Affinity DataIC50: 70nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328255(5-(2-chlorophenyl)-3-methyl-7-nitro-2,10-dihydrobe...)
Affinity DataIC50: 72nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328257(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 88nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328273(7-fluoro-3-methyl-5-phenyl-2,10-dihydrobenzo[e]pyr...)
Affinity DataIC50: 93nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328271(5-(2-chlorophenyl)-3-methyl-2,10-dihydrobenzo[e]py...)
Affinity DataIC50: 105nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328270(3-methyl-5-phenyl-2,10-dihydrobenzo[e]pyrazolo[4,3...)
Affinity DataIC50: 115nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328257(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 150nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328258(N-(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo...)
Affinity DataIC50: 180nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328277(7-chloro-5-(2-fluorophenyl)-2,10-dihydrobenzo[e]py...)
Affinity DataIC50: 190nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328265(5-(2-chlorophenyl)-7-nitro-3-phenyl-2,10-dihydrobe...)
Affinity DataIC50: 210nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328262(5-(2-chlorophenyl)-7-nitro-3-(trifluoromethyl)-2,1...)
Affinity DataIC50: 232nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328261((5-(2-chlorophenyl)-7-nitro-2,10-dihydrobenzo[e]py...)
Affinity DataIC50: 238nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328263(5-(2-chlorophenyl)-7-nitro-2,10-dihydrobenzo[e]pyr...)
Affinity DataIC50: 258nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328268(5-(2-chlorophenyl)-7-nitro-3-(pyridin-3-yl)-2,10-d...)
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328278(5-(2-chlorophenyl)-7-methoxy-2,10-dihydrobenzo[e]p...)
Affinity DataIC50: 320nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328276(7-chloro-5-(2-chlorophenyl)-2,10-dihydrobenzo[e]py...)
Affinity DataIC50: 440nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328275(7-chloro-5-phenyl-2,10-dihydrobenzo[e]pyrazolo[4,3...)
Affinity DataIC50: 490nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328258(N-(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo...)
Affinity DataIC50: 726nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328258(N-(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo...)
Affinity DataIC50: 930nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328257(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 989nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328256(5-(2-fluorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328257(5-(2-chlorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328259(6-(thiophen-2-yl)-4-(trifluoromethyl)-1H-pyrazolo[...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
LigandPNGBDBM50328266(5-(2-chlorophenyl)-7-nitro-3-phenethyl-2,10-dihydr...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of CDK2-cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328256(5-(2-fluorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328255(5-(2-chlorophenyl)-3-methyl-7-nitro-2,10-dihydrobe...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of FAKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328255(5-(2-chlorophenyl)-3-methyl-7-nitro-2,10-dihydrobe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328256(5-(2-fluorophenyl)-2,10-dihydrobenzo[e]pyrazolo[4,...)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50328255(5-(2-chlorophenyl)-3-methyl-7-nitro-2,10-dihydrobe...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed