Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50032185
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human 5HT2C receptor assessed as 10633-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human 5HT2B receptor assessed as 10633-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  384nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(N-butyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thiochrom...)
Affinity DataKi:  489nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi:  569nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(N-phenyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]is...)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(N-cyclohexyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-...)
Affinity DataKi:  1.77E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(N-o-tolyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]i...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi:  5.17E+3nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(N-propyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]is...)
Affinity DataKi:  6.60E+3nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Nisoxetine from human NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN-3542 from human DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(N-o-tolyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]i...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Citalopram from human SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325670(N-o-tolyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]i...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(N-butyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]iso...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(N-butyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]iso...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325669(N-butyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]iso...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(N-tert-butyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(N-tert-butyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325668(N-tert-butyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(N-cyclohexyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325659(8-fluoro-N-phenyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325667(N-cyclohexyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(N-propyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]is...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325666(N-propyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]is...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(N-isopropyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(N-isopropyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5HT2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325665(N-isopropyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(N-phenyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]is...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325664(N-phenyl-3,3a,4,9b-tetrahydro-1H-chromeno[4,3-c]is...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(N-butyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thiochrom...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325663(N-butyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thiochrom...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325662(N-cyclohexyl-8-fluoro-3,3a,4,9b-tetrahydro-1H-thio...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325661(8-fluoro-N-propyl-3,3a,4,9b-tetrahydro-1H-thiochro...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Csiro Molecular and Health Technologies

Curated by ChEMBL
LigandPNGBDBM50325660(8-fluoro-N-isopropyl-3,3a,4,9b-tetrahydro-1H-thioc...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Mesulergine from human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed