Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50032152
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324983(Cyclopropanecarboxylic acid[5-(3-methyl-[1,2,4]oxa...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324967(2-[(Furan-2-carbonyl)-amino]-4-phenyl-thiazole-5-c...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324975(N-[5-(5-Methyl-[1,2,4]oxadiazol-3-yl)-4-phenyl-thi...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324984(3-Methyl-N-[5-(3-methyl-[1,2,4]oxadiazol-5-yl)-4-p...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324972(Cyclopropanecarboxylic acid[5-(5-methyl-[1,2,4]oxa...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324973(3-Methyl-N-[5-(5-methyl-[1,2,4]oxadiazol-3-yl)-4-p...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324983(Cyclopropanecarboxylic acid[5-(3-methyl-[1,2,4]oxa...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324991(2-(3,4-Dimethoxy-phenyl)-N-[5-(2-ethyl-2H-tetrazol...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324984(3-Methyl-N-[5-(3-methyl-[1,2,4]oxadiazol-5-yl)-4-p...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324986(N-[5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-thi...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324968(Furan-2-carboxylic acid(5-butyryl-4-phenyl-thiazol...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324978(3-Methyl-N-(5-[1,2,4]oxadiazol-3-yl-4-phenyl-thiaz...)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324988(Cyclopropanecarboxylic acid[5-(2-ethyl-2H-tetrazol...)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324973(3-Methyl-N-[5-(5-methyl-[1,2,4]oxadiazol-3-yl)-4-p...)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324974(N-[5-(5-Methyl-[1,2,4]oxadiazol-3-yl)-4-phenyl-thi...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324968(Furan-2-carboxylic acid(5-butyryl-4-phenyl-thiazol...)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324969(Furan-2-carboxylic acid(5-ethoxymethyl-4-phenyl-th...)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324987(Furan-2-carboxylic acid[5-(2-ethyl-2H-tetrazol-5-y...)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324967(2-[(Furan-2-carbonyl)-amino]-4-phenyl-thiazole-5-c...)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324982(N-[5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-thi...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324977(Cyclopropanecarboxylic acid(5-[1,2,4]oxadiazol-3-y...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324972(Cyclopropanecarboxylic acid[5-(5-methyl-[1,2,4]oxa...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324985(N-[5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-thi...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324985(N-[5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-thi...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324971(N-[5-(5-Methyl-[1,2,4]oxadiazol-3-yl)-4-phenyl-thi...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324969(Furan-2-carboxylic acid(5-ethoxymethyl-4-phenyl-th...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324981(Furan-2-carboxylic acid[5-(3-methyl-[1,2,4]oxadiaz...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324988(Cyclopropanecarboxylic acid[5-(2-ethyl-2H-tetrazol...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324989(N-[5-(2-Ethyl-2H-tetrazol-5-yl)-4-phenyl-thiazol-2...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324976(Furan-2-carboxylic acid(5-[1,2,4]oxadiazol-3-yl-4-...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324975(N-[5-(5-Methyl-[1,2,4]oxadiazol-3-yl)-4-phenyl-thi...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324981(Furan-2-carboxylic acid[5-(3-methyl-[1,2,4]oxadiaz...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324992(Furan-2-carboxylic acid(5-cyano-4-phenyl-thiazol-2...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324979(N-(5-[1,2,4]Oxadiazol-3-yl-4-phenyl-thiazol-2-yl)-...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324977(Cyclopropanecarboxylic acid(5-[1,2,4]oxadiazol-3-y...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324979(N-(5-[1,2,4]Oxadiazol-3-yl-4-phenyl-thiazol-2-yl)-...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324978(3-Methyl-N-(5-[1,2,4]oxadiazol-3-yl-4-phenyl-thiaz...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324986(N-[5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-thi...)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324982(N-[5-(3-Methyl-[1,2,4]oxadiazol-5-yl)-4-phenyl-thi...)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324976(Furan-2-carboxylic acid(5-[1,2,4]oxadiazol-3-yl-4-...)
Affinity DataKi:  410nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324990(N-[5-(2-Ethyl-2H-tetrazol-5-yl)-4-phenyl-thiazol-2...)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324987(Furan-2-carboxylic acid[5-(2-ethyl-2H-tetrazol-5-y...)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324970(Furan-2-carboxylic acid[5-(5-methyl-[1,2,4]oxadiaz...)
Affinity DataKi:  700nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324980(N-(5-[1,2,4]Oxadiazol-3-yl-4-phenyl-thiazol-2-yl)-...)
Affinity DataKi:  710nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in buculovirus system by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324970(Furan-2-carboxylic acid[5-(5-methyl-[1,2,4]oxadiaz...)
Affinity DataKi:  780nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324990(N-[5-(2-Ethyl-2H-tetrazol-5-yl)-4-phenyl-thiazol-2...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Human)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50324991(2-(3,4-Dimethoxy-phenyl)-N-[5-(2-ethyl-2H-tetrazol...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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