Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50032080
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50272169(UFP-512 | H-Dmt-Tic-NH-(S)CH(CH2-COOH)-Bid | (S)-3...)
Affinity DataIC50: 0.120nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50179191(H-Dmt-Tic-NH-CH2-Bid | 2-[2-Amino-3-(4-hydroxy-2,6...)
Affinity DataIC50: 0.130nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324023((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataIC50: 0.320nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataIC50: 0.400nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50179191(H-Dmt-Tic-NH-CH2-Bid | 2-[2-Amino-3-(4-hydroxy-2,6...)
Affinity DataIC50: 26.9nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig small intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324023((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataIC50: 48.2nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig small intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324022((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataIC50: 50.1nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324021((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataIC50: 67.3nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50272169(UFP-512 | H-Dmt-Tic-NH-(S)CH(CH2-COOH)-Bid | (S)-3...)
Affinity DataIC50: 1.72E+3nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig small intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataIC50: 3.56E+3nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig small intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324022((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataIC50: 4.22E+3nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig small intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324021((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig small intestineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50179191(H-Dmt-Tic-NH-CH2-Bid | 2-[2-Amino-3-(4-hydroxy-2,6...)
Affinity DataKi:  0.0350nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324028((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-dime...)
Affinity DataKi:  0.118nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324023((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324019((S)-3-((S)-2-((S)-2-amino-3-(2,6-difluoro-4-hydrox...)
Affinity DataKi:  0.162nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324020((S)-3-((S)-2-((S)-2-amino-3-(4-hydroxyphenyl)propa...)
Affinity DataKi:  0.177nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataKi:  0.241nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324031(CHEMBL1214117 | N,N(CH3)2-Dmt-Tic-NH2 | (S)-2-((S)...)
Affinity DataKi:  0.309nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50272169(UFP-512 | H-Dmt-Tic-NH-(S)CH(CH2-COOH)-Bid | (S)-3...)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50179191(H-Dmt-Tic-NH-CH2-Bid | 2-[2-Amino-3-(4-hydroxy-2,6...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324025((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324022((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataKi:  0.913nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324021((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataKi:  1.01nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324023((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataKi:  1.68nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324025((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethy...)
Affinity DataKi:  4.05nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324029((S)-2-((S)-3-(2,6-difluoro-4-hydroxyphenyl)-2-(dim...)
Affinity DataKi:  29.2nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324030((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  34.8nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50272169(UFP-512 | H-Dmt-Tic-NH-(S)CH(CH2-COOH)-Bid | (S)-3...)
Affinity DataKi:  53.9nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324021((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataKi:  54.5nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324027((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxyphenyl)propa...)
Affinity DataKi:  63.9nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324022((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...)
Affinity DataKi:  66.9nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324026((S)-2-((S)-2-((S)-2-amino-3-(2,6-difluoro-4-hydrox...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324032((S)-2-((S)-3-(2,6-difluoro-4-hydroxyphenyl)-2-(dim...)
Affinity DataKi:  176nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324033((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  201nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324019((S)-3-((S)-2-((S)-2-amino-3-(2,6-difluoro-4-hydrox...)
Affinity DataKi:  225nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324031(CHEMBL1214117 | N,N(CH3)2-Dmt-Tic-NH2 | (S)-2-((S)...)
Affinity DataKi:  511nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324029((S)-2-((S)-3-(2,6-difluoro-4-hydroxyphenyl)-2-(dim...)
Affinity DataKi:  573nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324032((S)-2-((S)-3-(2,6-difluoro-4-hydroxyphenyl)-2-(dim...)
Affinity DataKi:  596nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324020((S)-3-((S)-2-((S)-2-amino-3-(4-hydroxyphenyl)propa...)
Affinity DataKi:  684nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324026((S)-2-((S)-2-((S)-2-amino-3-(2,6-difluoro-4-hydrox...)
Affinity DataKi:  1.03E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324030((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324033((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324027((S)-2-((S)-2-((S)-2-amino-3-(4-hydroxyphenyl)propa...)
Affinity DataKi:  1.65E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324028((S)-2-((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-dime...)
Affinity DataKi:  2.44E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed