Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50031967
TargetHistone deacetylase 1(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322419(Octanethioic acid S-[(E)-4-((5R,8S,11S)-5-benzyl-8...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322418(Octanethioic acid S-[(E)-4-((8S,11S)-8-isopropyl-6...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322422(Largazole | CHEMBL1173445)
Affinity DataIC50: 11.4nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322421(Octanethioic acid S-[(E)-4-((5R,8S,11S)-8-isopropy...)
Affinity DataIC50: 13.7nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 1(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322420(Octanethioic acid S-[(E)-4-((5R,8S,11S)-5-ethyl-8-...)
Affinity DataIC50: 161nMAssay Description:Inhibition of human recombinant HDAC1 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 4(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322418(Octanethioic acid S-[(E)-4-((8S,11S)-8-isopropyl-6...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 4(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322419(Octanethioic acid S-[(E)-4-((5R,8S,11S)-5-benzyl-8...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 4(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322422(Largazole | CHEMBL1173445)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 4(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322420(Octanethioic acid S-[(E)-4-((5R,8S,11S)-5-ethyl-8-...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 4(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 4(Human)
Universidade De Vigo

Curated by ChEMBL
LigandPNGBDBM50322421(Octanethioic acid S-[(E)-4-((5R,8S,11S)-8-isopropy...)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human recombinant HDAC4 after 15 mins by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed