Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50031830
LigandPNGBDBM50320097(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320098(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320101(N-(2-(dimethylamino)ethyl)-4-(3-(2-((7-fluoro-5-me...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320099(N-(2-(dimethylamino)ethyl)-4-(3-(2-((5-methoxy-2-(...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320101(N-(2-(dimethylamino)ethyl)-4-(3-(2-((7-fluoro-5-me...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320095(1-(2-((7-fluoro-5-methoxy-2-(1,3,5-trimethyl-1H-py...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320103(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320094(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320100(1-(2-((7-fluoro-5-methoxy-2-(1,3,5-trimethyl-1H-py...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320101(N-(2-(dimethylamino)ethyl)-4-(3-(2-((7-fluoro-5-me...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PI3deltaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320101(N-(2-(dimethylamino)ethyl)-4-(3-(2-((7-fluoro-5-me...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of PI3KbetaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320102(1-(2-((5-methoxy-1H-indol-3-yl)methylene)-3-oxo-2,...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320096(1-(2-((7-fluoro-5-methoxy-2-(1,3,5-trimethyl-1H-py...)
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320099(N-(2-(dimethylamino)ethyl)-4-(3-(2-((5-methoxy-2-(...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320103(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320096(1-(2-((7-fluoro-5-methoxy-2-(1,3,5-trimethyl-1H-py...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50320101(N-(2-(dimethylamino)ethyl)-4-(3-(2-((7-fluoro-5-me...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of PI3gammaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320095(1-(2-((7-fluoro-5-methoxy-2-(1,3,5-trimethyl-1H-py...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320100(1-(2-((7-fluoro-5-methoxy-2-(1,3,5-trimethyl-1H-py...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320098(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320097(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320094(1-(2-((5-methoxy-2-(1,3,5-trimethyl-1H-pyrazol-4-y...)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50320102(1-(2-((5-methoxy-1H-indol-3-yl)methylene)-3-oxo-2,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed