Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50031800
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266148(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319571(N-(4-(3-(2-((1-ethylpiperidin-4-yl)methylamino)pyr...)
Affinity DataIC50: 1nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266221(N-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]p...)
Affinity DataIC50: 2nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319572(N-(4-(3-(2-(2-(1-methylpyrrolidin-2-yl)ethylamino)...)
Affinity DataIC50: 2nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266149(1-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 5nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266148(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 9nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266185(N-[4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266187(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 16nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266148(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 19nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266149(1-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 23nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266187(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 25nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266185(N-[4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-...)
Affinity DataIC50: 27nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266221(N-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]p...)
Affinity DataIC50: 29nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
LigandPNGBDBM50266187(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 30nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
LigandPNGBDBM50266149(1-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 40nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266188(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 44nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319572(N-(4-(3-(2-(2-(1-methylpyrrolidin-2-yl)ethylamino)...)
Affinity DataIC50: 47nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266149(1-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 48nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
LigandPNGBDBM50319570(1-ethyl-3-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyr...)
Affinity DataIC50: 48nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266149(1-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 52nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319569(1-tert-butyl-3-(4-(3-(2-(methylamino)pyrimidin-4-y...)
Affinity DataIC50: 55nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266185(N-[4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-...)
Affinity DataIC50: 56nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
LigandPNGBDBM50266185(N-[4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-...)
Affinity DataIC50: 70nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266221(N-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]p...)
Affinity DataIC50: 77nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266188(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 80nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319573(N1-(4-(2-(4-(1H-benzo[d]imidazol-2-ylamino)naphtha...)
Affinity DataIC50: 82nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319574(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 86nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
LigandPNGBDBM50266188(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 88nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319571(N-(4-(3-(2-((1-ethylpiperidin-4-yl)methylamino)pyr...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319570(1-ethyl-3-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyr...)
Affinity DataIC50: 130nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266185(N-[4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-...)
Affinity DataIC50: 132nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266187(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 134nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266187(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 141nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266188(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 143nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319569(1-tert-butyl-3-(4-(3-(2-(methylamino)pyrimidin-4-y...)
Affinity DataIC50: 215nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319569(1-tert-butyl-3-(4-(3-(2-(methylamino)pyrimidin-4-y...)
Affinity DataIC50: 225nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319570(1-ethyl-3-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyr...)
Affinity DataIC50: 248nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319572(N-(4-(3-(2-(2-(1-methylpyrrolidin-2-yl)ethylamino)...)
Affinity DataIC50: 269nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266148(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 292nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319572(N-(4-(3-(2-(2-(1-methylpyrrolidin-2-yl)ethylamino)...)
Affinity DataIC50: 327nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319571(N-(4-(3-(2-((1-ethylpiperidin-4-yl)methylamino)pyr...)
Affinity DataIC50: 332nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266188(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 380nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319571(N-(4-(3-(2-((1-ethylpiperidin-4-yl)methylamino)pyr...)
Affinity DataIC50: 387nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50266221(N-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]p...)
Affinity DataIC50: 405nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319574(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 454nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319570(1-ethyl-3-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyr...)
Affinity DataIC50: 534nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319573(N1-(4-(2-(4-(1H-benzo[d]imidazol-2-ylamino)naphtha...)
Affinity DataIC50: 759nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319574(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
LigandPNGBDBM50266148(N-(4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-y...)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50319573(N1-(4-(2-(4-(1H-benzo[d]imidazol-2-ylamino)naphtha...)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
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