Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50031646
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316600(N,N-Dipropyl-[5-isothiocyanato-2-phenylindol-3-yl)...)
Affinity DataKd:  3.17nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316601(N,N-Dihexyl-[5-isothiocyanato-2-phenylindol-3-yl)g...)
Affinity DataKd:  5.07nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316602(N-(5-Isothiocyanato-2-phenylindol-3-ylglyoxyl)-N'-...)
Affinity DataKd:  8.31nMAssay Description:Irreversible binding affinity to TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316602(N-(5-Isothiocyanato-2-phenylindol-3-ylglyoxyl)-N'-...)
Affinity DataIC50: 42.2nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316600(N,N-Dipropyl-[5-isothiocyanato-2-phenylindol-3-yl)...)
Affinity DataIC50: 45.6nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316601(N,N-Dihexyl-[5-isothiocyanato-2-phenylindol-3-yl)g...)
Affinity DataIC50: 59.7nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316602(N-(5-Isothiocyanato-2-phenylindol-3-ylglyoxyl)-N'-...)
Affinity DataKi:  37.6nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316600(N,N-Dipropyl-[5-isothiocyanato-2-phenylindol-3-yl)...)
Affinity DataKi:  37.9nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50316601(N,N-Dihexyl-[5-isothiocyanato-2-phenylindol-3-yl)g...)
Affinity DataKi:  49.5nMAssay Description:Displacement of [3H]Ro5-4864 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed