Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50031779
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318963(rac-5-methyl-9-propyl-12-(tetrahydro-2H-pyran-2-yl...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318946(rac-9-(2-hydroxyethyl)-5-methyl-12-(tetrahydro-2H-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318959(rac-9-isobutyl-5-methyl-12-(tetrahydro-2H-pyran-2-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318960(rac-5-methyl-12-(tetrahydro-2H-pyran-2-yl)-5,7,8,9...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318958(rac-9-butyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 5nMAssay Description:Inhibition of VEGFR3 at 3 uMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318962(rac-9-ethyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318957(9-(2-hydroxyethyl)-6-methyl-12-(tetrahydro-2H-pyra...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318963(rac-5-methyl-9-propyl-12-(tetrahydro-2H-pyran-2-yl...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318949(6-methyl-12-(tetrahydro-2H-pyran-2-yl)-6,7,8,9-tet...)
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318951(9-ethyl-6-methyl-12-(tetrahydro-2H-pyran-2-yl)-6,7...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318970(rac-9-allyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318959(rac-9-isobutyl-5-methyl-12-(tetrahydro-2H-pyran-2-...)
Affinity DataIC50: 9nMAssay Description:Inhibition of VEGFR3 at 3 uMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318961(rac-5,9-dimethyl-12-(tetrahydro-2H-pyran-2-yl)-5,7...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318964(rac-9-isopropyl-5-methyl-12-(tetrahydro-2H-pyran-2...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318958(rac-9-butyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVECMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318958(rac-9-butyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318960(rac-5-methyl-12-(tetrahydro-2H-pyran-2-yl)-5,7,8,9...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318964(rac-9-isopropyl-5-methyl-12-(tetrahydro-2H-pyran-2...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318959(rac-9-isobutyl-5-methyl-12-(tetrahydro-2H-pyran-2-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVECMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318962(rac-9-ethyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVECMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318963(rac-5-methyl-9-propyl-12-(tetrahydro-2H-pyran-2-yl...)
Affinity DataIC50: 10nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVECMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318959(rac-9-isobutyl-5-methyl-12-(tetrahydro-2H-pyran-2-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318962(rac-9-ethyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318961(rac-5,9-dimethyl-12-(tetrahydro-2H-pyran-2-yl)-5,7...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318947(rac-9-(3-hydroxypropyl)-5-methyl-12-(tetrahydro-2H...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318948(rac-9-(2-(diethylamino)ethyl)-5-methyl-12-(tetrahy...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318959(rac-9-isobutyl-5-methyl-12-(tetrahydro-2H-pyran-2-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of VEGFR1 at 3 uMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318947(rac-9-(3-hydroxypropyl)-5-methyl-12-(tetrahydro-2H...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318945(rac-9-(2-ethoxyethyl)-5-methyl-12-(tetrahydro-2H-p...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318955(9-isobutyl-6-methyl-12-(tetrahydro-2H-pyran-2-yl)-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318970(rac-9-allyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318952(6-methyl-9-propyl-12-(tetrahydro-2H-pyran-2-yl)-6,...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318965(rac-9-isopentyl-5-methyl-12-(tetrahydro-2H-pyran-2...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318964(rac-9-isopropyl-5-methyl-12-(tetrahydro-2H-pyran-2...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318950(6,9-dimethyl-12-(tetrahydro-2H-pyran-2-yl)-6,7,8,9...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318945(rac-9-(2-ethoxyethyl)-5-methyl-12-(tetrahydro-2H-p...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318952(6-methyl-9-propyl-12-(tetrahydro-2H-pyran-2-yl)-6,...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318958(rac-9-butyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318946(rac-9-(2-hydroxyethyl)-5-methyl-12-(tetrahydro-2H-...)
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318958(rac-9-butyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 28nMAssay Description:Inhibition of VEGFR1 at 3 uMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318955(9-isobutyl-6-methyl-12-(tetrahydro-2H-pyran-2-yl)-...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318954(9-butyl-6-methyl-12-(tetrahydro-2H-pyran-2-yl)-6,7...)
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318961(rac-5,9-dimethyl-12-(tetrahydro-2H-pyran-2-yl)-5,7...)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318967(rac-9-cyclopentyl-5-methyl-12-(tetrahydro-2H-pyran...)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318968(rac-9-cyclohexyl-5-methyl-12-(tetrahydro-2H-pyran-...)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50318960(rac-5-methyl-12-(tetrahydro-2H-pyran-2-yl)-5,7,8,9...)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant TIE-2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318953(9-isopropyl-6-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 44nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318945(rac-9-(2-ethoxyethyl)-5-methyl-12-(tetrahydro-2H-p...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318970(rac-9-allyl-5-methyl-12-(tetrahydro-2H-pyran-2-yl)...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant VEGFR2 by time resolved fluorescence measurementsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318948(rac-9-(2-(diethylamino)ethyl)-5-methyl-12-(tetrahy...)
Affinity DataIC50: 50nMAssay Description:Inhibition of VEGF-stimulated VEGFR2 autophosphorylation in HUVECMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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