Report error Found 186 Enz. Inhib. hit(s) with all data for entry = 50031856
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 155nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 155nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 161nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 161nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 187nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 187nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 222nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 244nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 276nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 276nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 284nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 284nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Florida
Curated by ChEMBL
University of Florida
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 337nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 337nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in rat brain membrane after 3 hrsMore data for this Ligand-Target Pair
