Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 4629
LigandPNGBDBM81369(SW13)
Affinity DataIC50: 0.700nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81371(SW18)
Affinity DataIC50: 5nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81373(SW30)
Affinity DataIC50: 7nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50324735(CHEMBL568150 | AS605240 | (5E)-5-(QUINOXALIN-6-YLM...)
Affinity DataIC50: 8nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81370(SW14)
Affinity DataIC50: 9nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 11nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81368(PIK90)
Affinity DataIC50: 11nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81372(SW19)
Affinity DataIC50: 16nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81368(PIK90)
Affinity DataIC50: 18nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81370(SW14)
Affinity DataIC50: 21nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81369(SW13)
Affinity DataIC50: 33nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81371(SW18)
Affinity DataIC50: 38nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81368(PIK90)
Affinity DataIC50: 58nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50324735(CHEMBL568150 | AS605240 | (5E)-5-(QUINOXALIN-6-YLM...)
Affinity DataIC50: 60nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 162nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81369(SW13)
Affinity DataIC50: 221nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81367(PIK293)
Affinity DataIC50: 237nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50324735(CHEMBL568150 | AS605240 | (5E)-5-(QUINOXALIN-6-YLM...)
Affinity DataIC50: 270nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50324735(CHEMBL568150 | AS605240 | (5E)-5-(QUINOXALIN-6-YLM...)
Affinity DataIC50: 300nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81368(PIK90)
Affinity DataIC50: 350nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81372(SW19)
Affinity DataIC50: 376nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 486nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81370(SW14)
Affinity DataIC50: 697nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81373(SW30)
Affinity DataIC50: 740nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81369(SW13)
Affinity DataIC50: 1.24E+3nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81373(SW30)
Affinity DataIC50: 1.30E+3nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81371(SW18)
Affinity DataIC50: 2.40E+3nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81371(SW18)
Affinity DataIC50: 6.70E+3nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81372(SW19)
Affinity DataIC50: 7.90E+3nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81370(SW14)
Affinity DataIC50: 8.91E+3nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81367(PIK293)
Affinity DataIC50: 1.00E+4nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81373(SW30)
Affinity DataIC50: 8.50E+4nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM36411(PIK294 | CID24905149 | 2-((4-amino-3-(3-hydroxyphe...)
Affinity DataIC50: 9.00E+4nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81372(SW19)
Affinity DataIC50: 9.00E+4nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81367(PIK293)
Affinity DataIC50: 9.00E+4nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM81367(PIK293)
Affinity DataIC50: 9.00E+4nMAssay Description:Biochemical assay using PI3Ks and diversification of tolyl quinazolinone series.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed