Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50004347
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481978(CHEMBL1089622)
Affinity DataKd:  47nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481983(CHEMBL1089623)
Affinity DataKd:  48nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481980(CHEMBL1089627)
Affinity DataKd:  170nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481981(CHEMBL1089628)
Affinity DataKd:  980nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481984(CHEMBL1089626)
Affinity DataKd:  33nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481987(CHEMBL1089624)
Affinity DataKd:  920nMAssay Description:Binding affinity to human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by isothermal titration colorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481978(CHEMBL1089622)
Affinity DataIC50: 31nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481985(CHEMBL1089625)
Affinity DataIC50: 32nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481983(CHEMBL1089623)
Affinity DataIC50: 43nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481984(CHEMBL1089626)
Affinity DataIC50: 220nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481981(CHEMBL1089628)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481987(CHEMBL1089624)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481980(CHEMBL1089627)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481979(CHEMBL1076797)
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481986(CHEMBL1089954)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481982(CHEMBL1089955)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50481988(CHEMBL1089953)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human Pin1 S16A/Y23A mutant expressed in Escherichia coli BL21(DE3) by chymotrypsin-coupled PPIase inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed