Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50035951
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011913(CHEMBL286657 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 6.00E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011901(CHEMBL35650 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 6.50E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011899(CHEMBL35319 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 7.70E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011914(CHEMBL287460 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 7.80E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011904(CHEMBL435173 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 8.10E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011897(CHEMBL285513 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 8.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011902(CHEMBL288690 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 8.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011898(CHEMBL284630 | 2-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50: 8.70E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011905(CHEMBL285200 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50: 8.80E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011894(CHEMBL285687 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 8.90E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011912(CHEMBL35509 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 9.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011925(CHEMBL289459 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 9.30E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011920(CHEMBL35249 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 9.60E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011893(CHEMBL291015 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 9.60E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011896(CHEMBL286153 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50: 9.70E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011900(CHEMBL34605 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50: 9.90E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011924(CHEMBL34237 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 9.90E+4nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011922(CHEMBL287087 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 1.02E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011907(CHEMBL286078 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 1.04E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011919(CHEMBL35238 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 1.06E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011921(CHEMBL34670 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50: 1.09E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50031282(CHEBI:17630 | Kanamycin)
Affinity DataIC50: 1.10E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011906(CHEMBL287699 | Hexanoic acid {4-amino-6-[4,6-diami...)
Affinity DataIC50: 1.10E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011918(CHEMBL415861 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50: 1.15E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011895(CHEMBL285274 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 1.15E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011915(CHEMBL287846 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50: 1.16E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011917(CHEMBL290355 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 1.18E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011910(CHEMBL36133 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50: 1.20E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011923(CHEMBL34486 | N-{4-Amino-6-[4,6-diamino-3-(3-amino...)
Affinity DataIC50: 1.21E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011911(CHEMBL286825 | 5-amino-2-aminomethyl-6-[4,6-diamin...)
Affinity DataIC50: 1.23E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011909(CHEMBL416222 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50: 1.25E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011908(CHEMBL34525 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 1.29E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011892(CHEMBL35867 | 5-amino-2-aminomethyl-6-[4,6-diamino...)
Affinity DataIC50: 1.29E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50011916(CHEMBL285021 | N-{4-Amino-6-[4,6-diamino-3-(3-amin...)
Affinity DataIC50: 1.34E+5nMAssay Description:In vitro inhibition of lysosomal phospholipase activity for release of labeled lysophosphatidylcholineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/21/2012
Entry Details Article
PubMed