Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50001011
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50007838(CHEMBL160369 | 8-Cyclohexyl-1,3-dipropyl-3,7-dihyd...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82010(8-(4-Hydroxy-phenyl)-1,3-dipropyl-3,9-dihydro-puri...)
Affinity DataKi:  0.630nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011824(CHEMBL34004 | 8-Cyclopentyl-1-methyl-3-propyl-3,7-...)
Affinity DataKi:  0.850nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011842(CHEMBL284578 | 8-Cyclopentyl-3-methyl-1-propyl-3,7...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011838(CHEMBL32253 | 8-(4-Hydroxy-phenyl)-3-methyl-1-prop...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011835(CHEMBL416585 | 8-Cyclohexyl-1-methyl-3-propyl-3,7-...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011825(CHEMBL34504 | 1,3-Dipropyl-8-thiophen-3-yl-3,7-dih...)
Affinity DataKi:  2nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011836(CHEMBL34789 | 8-(4-Hydroxy-phenyl)-1-methyl-3-prop...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82025(8-Phenyl-1,3-dipropyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011841(CHEMBL33816 | 1,3-Dipropyl-8-pyridin-4-yl-3,7-dihy...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50005366(CHEMBL33722 | 1,3-Dipropyl-8-thiophen-2-yl-3,7-dih...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against Adenosine A1 receptor in rat cortex by displacement of [3H]-cyclohexyladenosine (CHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011833(CHEMBL33673 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-te...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011846(CHEMBL286347 | 1-Methyl-3-propyl-8-thiophen-3-yl-3...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity against Adenosine A1 receptor in rat cortex by displacement of [3H]-cyclohexyladenosine (CHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011839(CHEMBL285074 | 8-Cyclohexyl-3-methyl-1-propyl-3,7-...)
Affinity DataKi:  5nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011845(CHEMBL34784 | 4-(3-Methyl-2,6-dioxo-1-propyl-2,3,6...)
Affinity DataKi:  6nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011840(CHEMBL18887 | 1-Methyl-8-phenyl-3-propyl-3,7-dihyd...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011843(CHEMBL33169 | 3-Methyl-1-propyl-8-thiophen-3-yl-3,...)
Affinity DataKi:  6.40nMAssay Description:Binding affinity against Adenosine A1 receptor in rat cortex by displacement of [3H]-cyclohexyladenosine (CHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011834(CHEMBL428341 | 3-Methyl-8-phenyl-1-propyl-3,7-dihy...)
Affinity DataKi:  7nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011828(CHEMBL285865 | 1-Methyl-3-propyl-8-thiophen-2-yl-3...)
Affinity DataKi:  8.90nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011848(CHEMBL33893 | 3-Methyl-1-propyl-8-thiophen-2-yl-3,...)
Affinity DataKi:  9.70nMAssay Description:Binding affinity against Adenosine A1 receptor in rat cortex by displacement of [3H]-cyclohexyladenosine (CHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011849(CHEMBL287010 | 1,3-Dipropyl-8-pyridin-3-yl-3,7-dih...)
Affinity DataKi:  12nMAssay Description:Binding affinity against Adenosine A1 receptor in rat cortex by displacement of [3H]-cyclohexyladenosine (CHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011844(CHEMBL33611 | 4-(1-Methyl-2,6-dioxo-3-propyl-2,3,6...)
Affinity DataKi:  14nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50006713(CHEMBL283908 | 1,3-Dipropyl-8-styryl-3,7-dihydro-p...)
Affinity DataKi:  22nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011829(CHEMBL33762 | 1-Methyl-3-propyl-8-pyridin-4-yl-3,7...)
Affinity DataKi:  22nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011847(CHEMBL284825 | 3-Methyl-1-propyl-8-pyridin-4-yl-3,...)
Affinity DataKi:  28nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011830(CHEMBL33795 | 1-Methyl-3-propyl-8-styryl-3,7-dihyd...)
Affinity DataKi:  31nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011825(CHEMBL34504 | 1,3-Dipropyl-8-thiophen-3-yl-3,7-dih...)
Affinity DataKi:  39nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011830(CHEMBL33795 | 1-Methyl-3-propyl-8-styryl-3,7-dihyd...)
Affinity DataKi:  47nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011823(CHEMBL34120 | 3-Methyl-1-propyl-8-styryl-3,7-dihyd...)
Affinity DataKi:  50nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011823(CHEMBL34120 | 3-Methyl-1-propyl-8-styryl-3,7-dihyd...)
Affinity DataKi:  58nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50006697(CHEMBL33115 | 8-Phenethyl-1,3-dipropyl-3,7-dihydro...)
Affinity DataKi:  58nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  60nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82010(8-(4-Hydroxy-phenyl)-1,3-dipropyl-3,9-dihydro-puri...)
Affinity DataKi:  61nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011850(CHEMBL285212 | 3-Methyl-1-propyl-8-pyridin-3-yl-3,...)
Affinity DataKi:  70nMAssay Description:Binding affinity against Adenosine A1 receptor in rat cortex by displacement of [3H]-cyclohexyladenosine (CHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011846(CHEMBL286347 | 1-Methyl-3-propyl-8-thiophen-3-yl-3...)
Affinity DataKi:  70nMAssay Description:Binding affinity against Adenosine A2 receptor in rat striatum by displacement of [3H]N-ethyladenosine-5''-uronamide(NECA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011837(CHEMBL284598 | 1-Methyl-3-propyl-8-pyridin-3-yl-3,...)
Affinity DataKi:  73nMAssay Description:Binding affinity against Adenosine A1 receptor in rat cortex by displacement of [3H]-cyclohexyladenosine (CHA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011836(CHEMBL34789 | 8-(4-Hydroxy-phenyl)-1-methyl-3-prop...)
Affinity DataKi:  82nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50006713(CHEMBL283908 | 1,3-Dipropyl-8-styryl-3,7-dihydro-p...)
Affinity DataKi:  85nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011840(CHEMBL18887 | 1-Methyl-8-phenyl-3-propyl-3,7-dihyd...)
Affinity DataKi:  93nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM82025(8-Phenyl-1,3-dipropyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataKi:  116nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011841(CHEMBL33816 | 1,3-Dipropyl-8-pyridin-4-yl-3,7-dihy...)
Affinity DataKi:  136nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50005366(CHEMBL33722 | 1,3-Dipropyl-8-thiophen-2-yl-3,7-dih...)
Affinity DataKi:  173nMAssay Description:Binding affinity against Adenosine A2 receptor in rat striatum by displacement of [3H]N-ethyladenosine-5''-uronamide(NECA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011833(CHEMBL33673 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-te...)
Affinity DataKi:  189nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  230nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011824(CHEMBL34004 | 8-Cyclopentyl-1-methyl-3-propyl-3,7-...)
Affinity DataKi:  247nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011844(CHEMBL33611 | 4-(1-Methyl-2,6-dioxo-3-propyl-2,3,6...)
Affinity DataKi:  254nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011827(CHEMBL287011 | 1-Methyl-8-phenethyl-3-propyl-3,7-d...)
Affinity DataKi:  259nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011838(CHEMBL32253 | 8-(4-Hydroxy-phenyl)-3-methyl-1-prop...)
Affinity DataKi:  263nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by the displacement of [3H]N-ethyladenosine-5''-uronamide(NECA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50011831(CHEMBL32963 | 3-Methyl-8-phenethyl-1-propyl-3,7-di...)
Affinity DataKi:  275nMAssay Description:Binding affinity against adenosine A1 receptor in rat cortex by the displacement of [3H]cyclohexyladenosine (CHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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